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33332-25-1 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Mycobacterium kansasii
External ID: CHEMBL751698
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1996
Volume: 39
Issue: 17
First Page: 3394
Last Page: 3400
DOI: 10.1021/jm950538t

Target ChEMBL ID: CHEMBL614984
ChEMBL Target Name: Mycobacterium kansasii
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard Value
Log 1/MMIC=1.936
Log 1/MMIC=1.519
Log 1/MMIC=1.97
Log 1/MMIC=2.33
Log 1/MMIC=3.358
Log 1/MMIC=2.633
Log 1/MMIC=2.33
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Mycobacterium tuberculosis
External ID: CHEMBL750947
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1995
Volume: 38
Issue: 20
First Page: 3902
Last Page: 3907
DOI: 10.1021/jm00020a003

Target ChEMBL ID: CHEMBL360
ChEMBL Target Name: Mycobacterium tuberculosis
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=32ug.mL-1
MIC=16ug.mL-1
MIC=4ug.mL-1
MIC=1ug.mL-1
MIC<8ug.mL-1
MIC=0.25ug.mL-1
MIC=2ug.mL-1
MIC<0.03ug.mL-1
MIC=16ug.mL-1
MIC<8ug.mL-1
MIC=0.25ug.mL-1
MIC=2ug.mL-1
MIC=4ug.mL-1
MIC=64ug.mL-1
MIC=64ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Mycobacterium tuberculosis
External ID: CHEMBL750948
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1995
Volume: 38
Issue: 20
First Page: 3902
Last Page: 3907
DOI: 10.1021/jm00020a003

Target ChEMBL ID: CHEMBL360
ChEMBL Target Name: Mycobacterium tuberculosis
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=32ug.mL-1
MIC=32ug.mL-1
MIC=8ug.mL-1
MIC=2ug.mL-1
MIC=16ug.mL-1
MIC=0.5ug.mL-1
MIC=4ug.mL-1
MIC=1ug.mL-1
MIC=8ug.mL-1
MIC=16ug.mL-1
MIC=0.5ug.mL-1
MIC=0.25ug.mL-1
MIC=8ug.mL-1
MIC=64ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Mycobacterium kansasii
External ID: CHEMBL751696
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1995
Volume: 38
Issue: 20
First Page: 3902
Last Page: 3907
DOI: 10.1021/jm00020a003

Target ChEMBL ID: CHEMBL614984
ChEMBL Target Name: Mycobacterium kansasii
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=256ug.mL-1
MIC=2048ug.mL-1
MIC=2ug.mL-1
MIC=2ug.mL-1
MIC>64ug.mL-1
MIC<1ug.mL-1
MIC=8ug.mL-1
MIC=0.125ug.mL-1
MIC=32ug.mL-1
MIC>64ug.mL-1
MIC<1ug.mL-1
MIC<1ug.mL-1
MIC=8ug.mL-1
MIC=1024ug.mL-1
MIC=64ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Equus caballus
External ID: CHEMBL635957
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1996
Volume: 39
Issue: 17
First Page: 3394
Last Page: 3400
DOI: 10.1021/jm950538t

Target ChEMBL ID: CHEMBL613115
ChEMBL Target Name: Equus caballus
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
T1/2=2.8hr
T1/2=3.333hr
T1/2=1.833hr
T1/2=0.09167hr
T1/2=0.03833hr
T1/2=20hr
T1/2=0.1967hr
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Mycobacterium avium
External ID: CHEMBL749701
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1995
Volume: 38
Issue: 20
First Page: 3902
Last Page: 3907
DOI: 10.1021/jm00020a003

Target ChEMBL ID: CHEMBL614982
ChEMBL Target Name: Mycobacterium avium
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=64ug.mL-1
MIC=128ug.mL-1
MIC>256ug.mL-1
MIC=128ug.mL-1
MIC>64ug.mL-1
MIC=16ug.mL-1
MIC>256ug.mL-1
MIC>256ug.mL-1
MIC=128ug.mL-1
MIC=64ug.mL-1
MIC=64ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Mycobacterium avium
External ID: CHEMBL747038
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1995
Volume: 38
Issue: 20
First Page: 3902
Last Page: 3907
DOI: 10.1021/jm00020a003

Target ChEMBL ID: CHEMBL614982
ChEMBL Target Name: Mycobacterium avium
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC>1024ug.mL-1
MIC>2048ug.mL-1
MIC=256ug.mL-1
MIC=128ug.mL-1
MIC=256ug.mL-1
MIC=64ug.mL-1
MIC>64ug.mL-1
MIC=32ug.mL-1
MIC>256ug.mL-1
MIC=256ug.mL-1
MIC=128ug.mL-1
MIC=64ug.mL-1
MIC=64ug.mL-1
MIC=1024ug.mL-1
MIC>1024ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Mycobacterium tuberculosis
External ID: CHEMBL750950
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1995
Volume: 38
Issue: 20
First Page: 3902
Last Page: 3907
DOI: 10.1021/jm00020a003

Target ChEMBL ID: CHEMBL360
ChEMBL Target Name: Mycobacterium tuberculosis
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=32ug.mL-1
MIC=2048ug.mL-1
MIC=16ug.mL-1
MIC>16ug.mL-1
MIC=64ug.mL-1
MIC=0.5ug.mL-1
MIC<0.03ug.mL-1
MIC=64ug.mL-1
MIC=0.5ug.mL-1
MIC=2ug.mL-1
MIC>64ug.mL-1
MIC=64ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL636372
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1996
Volume: 39
Issue: 17
First Page: 3394
Last Page: 3400
DOI: 10.1021/jm950538t
Standard TypeStandard RelationStandard Value
LogP=0.67
LogP=0.91
LogP=1.19
LogP=2.21
LogP=4.98
LogP=1.7
LogP=1.97
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Mycobacterium tuberculosis
External ID: CHEMBL749416
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1996
Volume: 39
Issue: 17
First Page: 3394
Last Page: 3400
DOI: 10.1021/jm950538t

Target ChEMBL ID: CHEMBL360
ChEMBL Target Name: Mycobacterium tuberculosis
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard Value
Log 1/MMIC=1.635
Log 1/MMIC=1.218
Log 1/MMIC=2.271
Log 1/MMIC=2.934
Log 1/MMIC=3.977
Log 1/MMIC=1.73
Log 1/MMIC=2.031
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Mycobacterium tuberculosis
External ID: CHEMBL749417
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1996
Volume: 39
Issue: 17
First Page: 3394
Last Page: 3400
DOI: 10.1021/jm950538t

Target ChEMBL ID: CHEMBL360
ChEMBL Target Name: Mycobacterium tuberculosis
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard Value
Log 1/MMIC=1.334
Log 1/MMIC=1.218
Log 1/MMIC=1.97
Log 1/MMIC=3.633
Log 1/MMIC=2.455
Log 1/MMIC=2.031
Log 1/MMIC=2.934
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Mycobacterium avium
External ID: CHEMBL882186
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1996
Volume: 39
Issue: 17
First Page: 3394
Last Page: 3400
DOI: 10.1021/jm950538t

Target ChEMBL ID: CHEMBL614982
ChEMBL Target Name: Mycobacterium avium
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard Value
Log 1/MMIC=0.431
Log 1/MMIC=0.013
Log 1/MMIC=0.164
Log 1/MMIC=0.225
Log 1/MMIC=1.25
Log 1/MMIC=2.33
Log 1/MMIC=0.526
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Mycobacterium tuberculosis
External ID: CHEMBL749418
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1996
Volume: 39
Issue: 17
First Page: 3394
Last Page: 3400
DOI: 10.1021/jm950538t

Target ChEMBL ID: CHEMBL360
ChEMBL Target Name: Mycobacterium tuberculosis
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard Value
Log 1/MMIC=1.033
Log 1/MMIC=1.218
Log 1/MMIC=1.067
Log 1/MMIC=2.633
Log 1/MMIC=3.977
Log 1/MMIC=1.73
Log 1/MMIC=2.031
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Mycobacterium avium
External ID: CHEMBL745305
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1996
Volume: 39
Issue: 17
First Page: 3394
Last Page: 3400
DOI: 10.1021/jm950538t

Target ChEMBL ID: CHEMBL614982
ChEMBL Target Name: Mycobacterium avium
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard Value
Log 1/MMIC=-0.071
Log 1/MMIC=0.013
Log 1/MMIC=0.164
Log 1/MMIC=0.526
Log 1/MMIC=0.949
Log 1/MMIC=0.225
Log 1/MMIC=0.526