| Standard Type | Standard Relation | Standard Value | Standard Units |
|---|---|---|---|
| Inhibition | = | 67.1 | % |
| Inhibition | = | 52.7 | % |
| Inhibition | = | 49.1 | % |
| Inhibition | = | 60 | % |
| Inhibition | = | 27.4 | % |
| Inhibition | = | 54.5 | % |
| Inhibition | = | 69.6 | % |
| Inhibition | = | 45.3 | % |
| Inhibition | = | 66 | % |
| Inhibition | = | 50.1 | % |
| Standard Type | Standard Relation | Standard Value |
|---|---|---|
| LogP | = | 4.02 |
| LogP | = | 4.14 |
| LogP | = | 2.96 |
| LogP | = | 4.07 |
| LogP | = | 5.4 |
| LogP | = | 5.25 |
| LogP | = | 4.07 |
| LogP | = | 1.21 |
| LogP | = | 3.68 |
| LogP | = | 5.79 |
| LogP | = | 8.96 |
| LogP | = | 3.7 |
| LogP | = | 4.21 |
| LogP | = | 3.98 |
| LogP | = | 4.4 |
| LogP | = | 3.57 |
| LogP | = | 4.19 |
| LogP | = | 3.59 |
| LogP | = | 5.65 |
| LogP | = | 6.13 |
| PubChem Standard Value | Standard Type | Standard Relation | Standard Value | Standard Units | Data Validity Comment |
|---|---|---|---|---|---|
| 3.98107 | IC50 | = | 3981.07 | nM | |
| 3.63078 | IC50 | = | 3630.78 | nM | |
| 7.07946 | IC50 | = | 7079.46 | nM | |
| 3.23594 | IC50 | = | 3235.94 | nM | |
| 1.62181 | IC50 | = | 1621.81 | nM | |
| 17.378 | IC50 | = | 17378.01 | nM | |
| 2.13796 | IC50 | = | 2137.96 | nM | |
| 2.88403 | IC50 | = | 2884.03 | nM | |
| 128.825 | IC50 | = | 128824.96 | nM | Outside typical range |
| 2.04174 | IC50 | = | 2041.74 | nM | |
| 4.89779 | IC50 | = | 4897.79 | nM | |
| 2.69153 | IC50 | = | 2691.53 | nM | |
| 1.94984 | IC50 | = | 1949.84 | nM | |
| 602.56 | IC50 | = | 602559.59 | nM | Outside typical range |
| 10.9648 | IC50 | = | 10964.78 | nM | |
| 22.3872 | IC50 | = | 22387.21 | nM | |
| 301.995 | IC50 | = | 301995.17 | nM | Outside typical range |
| 3.54813 | IC50 | = | 3548.13 | nM | |
| 1.23027 | IC50 | = | 1230.27 | nM | |
| 1000 | IC50 | > | 1000000 | nM | Outside typical range |
| Standard Type | Standard Relation | Standard Value | Standard Units |
|---|---|---|---|
| Inhibition | = | 25.8 | % |
| Inhibition | = | 58.7 | % |
| Inhibition | = | 39.7 | % |
| Inhibition | = | 47.8 | % |
| Inhibition | = | 33.6 | % |
| Inhibition | = | 56.2 | % |
| Inhibition | = | 56.8 | % |
| Inhibition | = | 39 | % |
| PubChem Standard Value | Standard Type | Standard Relation | Standard Value | Standard Units | Data Validity Comment |
|---|---|---|---|---|---|
| 0.43652 | IC50 | = | 436.52 | nM | |
| 1.25893 | IC50 | = | 1258.93 | nM | |
| 1.23027 | IC50 | = | 1230.27 | nM | |
| 1.09648 | IC50 | = | 1096.48 | nM | |
| 891.251 | IC50 | = | 891250.94 | nM | Outside typical range |
| 7.07946 | IC50 | = | 7079.46 | nM | |
| 1.65959 | IC50 | = | 1659.59 | nM | |
| 0.18621 | IC50 | = | 186.21 | nM | |
| 1.90546 | IC50 | = | 1905.46 | nM | |
| 9.12011 | IC50 | = | 9120.11 | nM | |
| 1.20226 | IC50 | = | 1202.26 | nM | |
| 0.33113 | IC50 | = | 331.13 | nM | |
| 0.95499 | IC50 | = | 954.99 | nM | |
| 0.21878 | IC50 | = | 218.78 | nM | |
| 0.6166 | IC50 | = | 616.6 | nM | |
| 45.7088 | IC50 | = | 45708.82 | nM | |
| 3.01995 | IC50 | = | 3019.95 | nM | |
| 0.58884 | IC50 | = | 588.84 | nM | |
| 1.99526 | IC50 | = | 1995.26 | nM | |
| 0.37154 | IC50 | = | 371.54 | nM |