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3033-80-5 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:T47D
External ID: CHEMBL2329264
Protocol: N/A
Comment: Journal: ACS Med. Chem. Lett.
Year: 2013
Volume: 4
Issue: 2
First Page: 170
Last Page: 174
DOI: 10.1021/ml300238z

Target ChEMBL ID: CHEMBL614361
ChEMBL Target Name: T47D
ChEMBL Target Type: CELL-LINE - Target is a specific cell-line
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
Activity=52.6%
Activity=46.54%
Activity=72.92%
Activity=37.92%
Activity=63.43%
Activity=8.37%
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:K562
External ID: CHEMBL2329263
Protocol: N/A
Comment: Journal: ACS Med. Chem. Lett.
Year: 2013
Volume: 4
Issue: 2
First Page: 170
Last Page: 174
DOI: 10.1021/ml300238z

Target ChEMBL ID: CHEMBL385
ChEMBL Target Name: K562
ChEMBL Target Type: CELL-LINE - Target is a specific cell-line
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
Activity=26.66%
Activity=34.46%
Activity=23.08%
Activity=27.15%
Activity=21.38%
Activity=7%
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Escherichia coli
External ID: CHEMBL3101599
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 2014
Volume: 24
Issue: 1
First Page: 367
Last Page: 370
DOI: 10.1016/j.bmcl.2013.10.072

Target ChEMBL ID: CHEMBL354
ChEMBL Target Name: Escherichia coli
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=7.5ug.mL-1
MIC>50ug.mL-1
MIC>50ug.mL-1
MIC>50ug.mL-1
MIC>50ug.mL-1
MIC>50ug.mL-1
MIC>50ug.mL-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Staphylococcus aureus
External ID: CHEMBL3101600
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 2014
Volume: 24
Issue: 1
First Page: 367
Last Page: 370
DOI: 10.1016/j.bmcl.2013.10.072

Target ChEMBL ID: CHEMBL352
ChEMBL Target Name: Staphylococcus aureus
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=3.125ug.mL-1
MIC=6.25ug.mL-1
MIC>50ug.mL-1
MIC>50ug.mL-1
MIC=50ug.mL-1
MIC>50ug.mL-1
MIC=50ug.mL-1