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288-14-2 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL623554
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 1998
Volume: 8
Issue: 9
First Page: 1113
Last Page: 1116
DOI: 10.1016/s0960-894x(98)00165-6
Standard TypeStandard RelationStandard ValueStandard Units
(kcat/KM)/kuncat=3600000M-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL2173908
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 2012
Volume: 55
Issue: 13
First Page: 6002
Last Page: 6020
DOI: 10.1021/jm300343m
Standard TypeStandard RelationStandard Value
pKa=-2.97
pKa=5.2
pKa=7
pKa=2.19
pKa=2.3
pKa=2.52
pKa=-3.8
pKa=1.3
pKa=0.4
pKa=11.2
pKa=8.4
pKa=11.27
pKa=9.8
pKa=0.8
pKa=-5
pKa=10.7
pKa=10.89
pKa=-0.51