HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Proto-oncogene tyrosine-protein kinase receptor Ret

External ID: CHEMBL5054531

Protocol: N/A

Comment: Journal: Bioorg Med Chem
Year: 2021
Volume: 48
First Page: 116422
Last Page: 116422
DOI: 10.1016/j.bmc.2021.116422

Target ChEMBL ID: CHEMBL2041
ChEMBL Target Name: Tyrosine-protein kinase receptor RET
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

Standard Type	Standard Relation	Standard Value	Standard Units
Inhibition	=	17.8	%

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Platelet-derived growth factor receptor beta

External ID: CHEMBL5054530

Protocol: N/A

Comment: Journal: Bioorg Med Chem
Year: 2021
Volume: 48
First Page: 116422
Last Page: 116422
DOI: 10.1016/j.bmc.2021.116422

Target ChEMBL ID: CHEMBL1913
ChEMBL Target Name: Platelet-derived growth factor receptor beta
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

Standard Type	Standard Relation	Standard Value	Standard Units
Inhibition	=	26	%

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Platelet-derived growth factor receptor alpha

External ID: CHEMBL5054529

Protocol: N/A

Comment: Journal: Bioorg Med Chem
Year: 2021
Volume: 48
First Page: 116422
Last Page: 116422
DOI: 10.1016/j.bmc.2021.116422

Target ChEMBL ID: CHEMBL2007
ChEMBL Target Name: Platelet-derived growth factor receptor alpha
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

Standard Type	Standard Relation	Standard Value	Standard Units
Inhibition	=	81.8	%

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Vascular endothelial growth factor receptor 3

External ID: CHEMBL5054528

Protocol: N/A

Comment: Journal: Bioorg Med Chem
Year: 2021
Volume: 48
First Page: 116422
Last Page: 116422
DOI: 10.1016/j.bmc.2021.116422

Target ChEMBL ID: CHEMBL1955
ChEMBL Target Name: Vascular endothelial growth factor receptor 3
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

Standard Type	Standard Relation	Standard Value	Standard Units
Inhibition	=	4.6	%

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Receptor tyrosine-protein kinase erbB-4

External ID: CHEMBL5054535

Protocol: N/A

Comment: Journal: Bioorg Med Chem
Year: 2021
Volume: 48
First Page: 116422
Last Page: 116422
DOI: 10.1016/j.bmc.2021.116422

Target ChEMBL ID: CHEMBL3009
ChEMBL Target Name: Receptor protein-tyrosine kinase erbB-4
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

Standard Type	Standard Relation	Standard Value	Standard Units
Inhibition	=	14.4	%

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Receptor tyrosine-protein kinase erbB-2

External ID: CHEMBL5054534

Protocol: N/A

Comment: Journal: Bioorg Med Chem
Year: 2021
Volume: 48
First Page: 116422
Last Page: 116422
DOI: 10.1016/j.bmc.2021.116422

Target ChEMBL ID: CHEMBL1824
ChEMBL Target Name: Receptor protein-tyrosine kinase erbB-2
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

Standard Type	Standard Relation	Standard Value	Standard Units
Inhibition	=	31.5	%

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Epidermal growth factor receptor

External ID: CHEMBL5054533

Protocol: N/A

Comment: Journal: Bioorg Med Chem
Year: 2021
Volume: 48
First Page: 116422
Last Page: 116422
DOI: 10.1016/j.bmc.2021.116422

Target ChEMBL ID: CHEMBL203
ChEMBL Target Name: Epidermal growth factor receptor erbB1
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

Standard Type	Standard Relation	Standard Value	Standard Units
Inhibition	=	10.8	%

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Mast/stem cell growth factor receptor Kit

External ID: CHEMBL5054532

Protocol: N/A

Comment: Journal: Bioorg Med Chem
Year: 2021
Volume: 48
First Page: 116422
Last Page: 116422
DOI: 10.1016/j.bmc.2021.116422

Target ChEMBL ID: CHEMBL1936
ChEMBL Target Name: Stem cell growth factor receptor
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

Standard Type	Standard Relation	Standard Value	Standard Units
Inhibition	=	94.4	%

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：MOLM-13

External ID: CHEMBL5054521

Protocol: N/A

Comment: Compounds with activity <= 10uM or explicitly reported as active by ChEMBL are flagged as active in this PubChem assay presentation.

Journal: Bioorg Med Chem
Year: 2021
Volume: 48
First Page: 116422
Last Page: 116422
DOI: 10.1016/j.bmc.2021.116422

Target ChEMBL ID: CHEMBL3706572
ChEMBL Target Name: MOLM-13
ChEMBL Target Type: CELL-LINE - Target is a specific cell-line
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular

PubChem Standard Value	Standard Type	Standard Relation	Standard Value	Standard Units
0.0283	IC50	=	28.3	nM
0.0194	IC50	=	19.4	nM
1	IC50	>	1000	nM

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Receptor-type tyrosine-protein kinase FLT3

External ID: CHEMBL5054520

Protocol: N/A

Comment: Compounds with activity <= 10uM or explicitly reported as active by ChEMBL are flagged as active in this PubChem assay presentation.

Journal: Bioorg Med Chem
Year: 2021
Volume: 48
First Page: 116422
Last Page: 116422
DOI: 10.1016/j.bmc.2021.116422

Target ChEMBL ID: CHEMBL1974
ChEMBL Target Name: Tyrosine-protein kinase receptor FLT3
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

PubChem Standard Value	Standard Type	Standard Relation	Standard Value	Standard Units
0.0013	IC50	=	1.3	nM
0.1441	IC50	=	144.1	nM
0.0072	IC50	=	7.2	nM

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Vascular endothelial growth factor receptor 2

External ID: CHEMBL5054527

Protocol: N/A

Comment: Journal: Bioorg Med Chem
Year: 2021
Volume: 48
First Page: 116422
Last Page: 116422
DOI: 10.1016/j.bmc.2021.116422

Target ChEMBL ID: CHEMBL279
ChEMBL Target Name: Vascular endothelial growth factor receptor 2
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

Standard Type	Standard Relation	Standard Value	Standard Units
Inhibition	=	9.7	%

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Vascular endothelial growth factor receptor 1

External ID: CHEMBL5054526

Protocol: N/A

Comment: Journal: Bioorg Med Chem
Year: 2021
Volume: 48
First Page: 116422
Last Page: 116422
DOI: 10.1016/j.bmc.2021.116422

Target ChEMBL ID: CHEMBL1868
ChEMBL Target Name: Vascular endothelial growth factor receptor 1
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

Standard Type	Standard Relation	Standard Value	Standard Units
Inhibition	=	3.6	%

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Receptor-type tyrosine-protein kinase FLT3

External ID: CHEMBL5054525

Protocol: N/A

Comment: Journal: Bioorg Med Chem
Year: 2021
Volume: 48
First Page: 116422
Last Page: 116422
DOI: 10.1016/j.bmc.2021.116422

Target ChEMBL ID: CHEMBL1974
ChEMBL Target Name: Tyrosine-protein kinase receptor FLT3
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

Standard Type	Standard Relation	Standard Value	Standard Units
Inhibition	=	99.2	%

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Receptor-type tyrosine-protein kinase FLT3

External ID: CHEMBL5054519

Protocol: N/A

Comment: Compounds with activity <= 10uM or explicitly reported as active by ChEMBL are flagged as active in this PubChem assay presentation.

Journal: Bioorg Med Chem
Year: 2021
Volume: 48
First Page: 116422
Last Page: 116422
DOI: 10.1016/j.bmc.2021.116422

Target ChEMBL ID: CHEMBL1974
ChEMBL Target Name: Tyrosine-protein kinase receptor FLT3
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

PubChem Standard Value	Standard Type	Standard Relation	Standard Value	Standard Units
0.0035	IC50	=	3.5	nM
0.0382	IC50	=	38.2	nM
0.0087	IC50	=	8.7	nM

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：MV4-11

External ID: CHEMBL5054518

Protocol: N/A

Comment: Compounds with activity <= 10uM or explicitly reported as active by ChEMBL are flagged as active in this PubChem assay presentation.

Journal: Bioorg Med Chem
Year: 2021
Volume: 48
First Page: 116422
Last Page: 116422
DOI: 10.1016/j.bmc.2021.116422

Target ChEMBL ID: CHEMBL613835
ChEMBL Target Name: MV4-11
ChEMBL Target Type: CELL-LINE - Target is a specific cell-line
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular

PubChem Standard Value	Standard Type	Standard Relation	Standard Value	Standard Units
0.0112	IC50	=	11.2	nM
0.0053	IC50	=	5.3	nM
0.1725	IC50	=	172.5	nM

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Tyrosine-protein kinase ITK/TSK

External ID: CHEMBL5054547

Protocol: N/A

Comment: Journal: Bioorg Med Chem
Year: 2021
Volume: 48
First Page: 116422
Last Page: 116422
DOI: 10.1016/j.bmc.2021.116422

Target ChEMBL ID: CHEMBL2959
ChEMBL Target Name: Tyrosine-protein kinase ITK/TSK
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

Standard Type	Standard Relation	Standard Value	Standard Units
Inhibition	=	32	%

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Focal adhesion kinase 1

External ID: CHEMBL5054546

Protocol: N/A

Comment: Journal: Bioorg Med Chem
Year: 2021
Volume: 48
First Page: 116422
Last Page: 116422
DOI: 10.1016/j.bmc.2021.116422

Target ChEMBL ID: CHEMBL2695
ChEMBL Target Name: Focal adhesion kinase 1
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

Standard Type	Standard Relation	Standard Value	Standard Units
Inhibition	=	34.8	%

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Activated CDC42 kinase 1

External ID: CHEMBL5054545

Protocol: N/A

Comment: Journal: Bioorg Med Chem
Year: 2021
Volume: 48
First Page: 116422
Last Page: 116422
DOI: 10.1016/j.bmc.2021.116422

Target ChEMBL ID: CHEMBL4599
ChEMBL Target Name: Tyrosine kinase non-receptor protein 2
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

Standard Type	Standard Relation	Standard Value	Standard Units
Inhibition	=	15.2	%

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Tyrosine-protein kinase BTK

External ID: CHEMBL5054544

Protocol: N/A

Comment: Journal: Bioorg Med Chem
Year: 2021
Volume: 48
First Page: 116422
Last Page: 116422
DOI: 10.1016/j.bmc.2021.116422

Target ChEMBL ID: CHEMBL5251
ChEMBL Target Name: Tyrosine-protein kinase BTK
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

Standard Type	Standard Relation	Standard Value	Standard Units
Inhibition	=	6.2	%

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Insulin receptor

External ID: CHEMBL5054550

Protocol: N/A

Comment: Journal: Bioorg Med Chem
Year: 2021
Volume: 48
First Page: 116422
Last Page: 116422
DOI: 10.1016/j.bmc.2021.116422

Target ChEMBL ID: CHEMBL1981
ChEMBL Target Name: Insulin receptor
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

Standard Type	Standard Relation	Standard Value	Standard Units
Inhibition	=	63.3	%

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Receptor-type tyrosine-protein kinase FLT3

External ID: CHEMBL5054549

Protocol: N/A

Comment: Journal: Bioorg Med Chem
Year: 2021
Volume: 48
First Page: 116422
Last Page: 116422
DOI: 10.1016/j.bmc.2021.116422

Target ChEMBL ID: CHEMBL1974
ChEMBL Target Name: Tyrosine-protein kinase receptor FLT3
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

Standard Type	Standard Relation	Standard Value	Standard Units
Inhibition	=	100	%
Inhibition	=	100	%

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Receptor-type tyrosine-protein kinase FLT3

External ID: CHEMBL5054548

Protocol: N/A

Comment: Journal: Bioorg Med Chem
Year: 2021
Volume: 48
First Page: 116422
Last Page: 116422
DOI: 10.1016/j.bmc.2021.116422

Target ChEMBL ID: CHEMBL1974
ChEMBL Target Name: Tyrosine-protein kinase receptor FLT3
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

Standard Type	Standard Relation	Standard Value	Standard Units
Inhibition	=	100	%
Inhibition	=	100	%

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Insulin-like growth factor 1 receptor

External ID: CHEMBL5054539

Protocol: N/A

Comment: Journal: Bioorg Med Chem
Year: 2021
Volume: 48
First Page: 116422
Last Page: 116422
DOI: 10.1016/j.bmc.2021.116422

Target ChEMBL ID: CHEMBL1957
ChEMBL Target Name: Insulin-like growth factor I receptor
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

Standard Type	Standard Relation	Standard Value	Standard Units
Inhibition	=	54.9	%

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Ephrin type-A receptor 2

External ID: CHEMBL5054538

Protocol: N/A

Comment: Journal: Bioorg Med Chem
Year: 2021
Volume: 48
First Page: 116422
Last Page: 116422
DOI: 10.1016/j.bmc.2021.116422

Target ChEMBL ID: CHEMBL2068
ChEMBL Target Name: Ephrin type-A receptor 2
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

Standard Type	Standard Relation	Standard Value	Standard Units
Inhibition	=	9.7	%

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Tyrosine-protein kinase ABL1

External ID: CHEMBL5054537

Protocol: N/A

Comment: Journal: Bioorg Med Chem
Year: 2021
Volume: 48
First Page: 116422
Last Page: 116422
DOI: 10.1016/j.bmc.2021.116422

Target ChEMBL ID: CHEMBL1862
ChEMBL Target Name: Tyrosine-protein kinase ABL
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

Standard Type	Standard Relation	Standard Value	Standard Units
Inhibition	=	1.5	%

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Proto-oncogene tyrosine-protein kinase Src

External ID: CHEMBL5054536

Protocol: N/A

Comment: Journal: Bioorg Med Chem
Year: 2021
Volume: 48
First Page: 116422
Last Page: 116422
DOI: 10.1016/j.bmc.2021.116422

Target ChEMBL ID: CHEMBL267
ChEMBL Target Name: Tyrosine-protein kinase SRC
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

Standard Type	Standard Relation	Standard Value	Standard Units
Inhibition	=	10.4	%

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Fibroblast growth factor receptor 4

External ID: CHEMBL5054543

Protocol: N/A

Comment: Journal: Bioorg Med Chem
Year: 2021
Volume: 48
First Page: 116422
Last Page: 116422
DOI: 10.1016/j.bmc.2021.116422

Target ChEMBL ID: CHEMBL3973
ChEMBL Target Name: Fibroblast growth factor receptor 4
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

Standard Type	Standard Relation	Standard Value	Standard Units
Inhibition	=	31.6	%

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Fibroblast growth factor receptor 3

External ID: CHEMBL5054542

Protocol: N/A

Comment: Journal: Bioorg Med Chem
Year: 2021
Volume: 48
First Page: 116422
Last Page: 116422
DOI: 10.1016/j.bmc.2021.116422

Target ChEMBL ID: CHEMBL2742
ChEMBL Target Name: Fibroblast growth factor receptor 3
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

Standard Type	Standard Relation	Standard Value	Standard Units
Inhibition	=	0	%

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Fibroblast growth factor receptor 2

External ID: CHEMBL5054541

Protocol: N/A

Comment: Journal: Bioorg Med Chem
Year: 2021
Volume: 48
First Page: 116422
Last Page: 116422
DOI: 10.1016/j.bmc.2021.116422

Target ChEMBL ID: CHEMBL4142
ChEMBL Target Name: Fibroblast growth factor receptor 2
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

Standard Type	Standard Relation	Standard Value	Standard Units
Inhibition	=	41.8	%

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Fibroblast growth factor receptor 1

External ID: CHEMBL5054540

Protocol: N/A

Comment: Journal: Bioorg Med Chem
Year: 2021
Volume: 48
First Page: 116422
Last Page: 116422
DOI: 10.1016/j.bmc.2021.116422

Target ChEMBL ID: CHEMBL3650
ChEMBL Target Name: Fibroblast growth factor receptor 1
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

Standard Type	Standard Relation	Standard Value	Standard Units
Inhibition	=	12.2	%

2489446-47-9 靶点实验数据