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2139-03-9 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Putative dihydropicolinate synthase
External ID: CHEMBL669832
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 1994
Volume: 4
Issue: 19
First Page: 2267
Last Page: 2272
DOI: 10.1016/0960-894X(94)85023-2

Target ChEMBL ID: CHEMBL3430
ChEMBL Target Name: Dihydrodipicolinate synthase
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: H - Homologous protein target assigned
Confidence: Homologous single protein target assigned
Standard TypeStandard RelationStandard ValueStandard Units
Inhibition=43%
Inhibition=0%
Inhibition=0%
Inhibition=0%
Inhibition=0%
Inhibition=0%
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL633002
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 1993
Volume: 3
Issue: 6
First Page: 1193
Last Page: 1196
DOI: 10.1016/S0960-894X(00)80313-3
Standard TypeStandard RelationStandard Value
pKa=1.8
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL633003
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 1993
Volume: 3
Issue: 6
First Page: 1193
Last Page: 1196
DOI: 10.1016/S0960-894X(00)80313-3
Standard TypeStandard RelationStandard Value
pKa=6.2