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19084-26-5 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Mycobacterium tuberculosis
External ID: CHEMBL3377978
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 2014
Volume: 24
Issue: 14
First Page: 3118
Last Page: 3120
DOI: 10.1016/j.bmcl.2014.05.006

Target ChEMBL ID: CHEMBL360
ChEMBL Target Name: Mycobacterium tuberculosis
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard UnitsActivity Comment
MIC=0.7ug.mL-1
MIC=1.5ug.mL-1
MICNot Determined
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Mus musculus
External ID: CHEMBL3377979
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 2014
Volume: 24
Issue: 14
First Page: 3118
Last Page: 3120
DOI: 10.1016/j.bmcl.2014.05.006

Target ChEMBL ID: CHEMBL375
ChEMBL Target Name: Mus musculus
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard UnitsActivity Comment
LD50=133mg.kg-1
LD50=315mg.kg-1
LD50=405mg.kg-1
LD50Not Determined
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Mycobacterium avium
External ID: CHEMBL3377976
Protocol: N/A
Comment: Journal: Bioorg. Med. Chem. Lett.
Year: 2014
Volume: 24
Issue: 14
First Page: 3118
Last Page: 3120
DOI: 10.1016/j.bmcl.2014.05.006

Target ChEMBL ID: CHEMBL614982
ChEMBL Target Name: Mycobacterium avium
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard UnitsActivity Comment
MIC=0.1ug.mL-1
MICNot Determined
MIC=0.3ug.mL-1
MIC=0.7ug.mL-1
MICNot Determined
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Mycolicibacter terrae
External ID: CHEMBL3377977
Protocol: N/A
Comment: Journal: Bioorg Med Chem Lett
Year: 2014
Volume: 24
Issue: 14
First Page: 3118
Last Page: 3120
DOI: 10.1016/j.bmcl.2014.05.006

Target ChEMBL ID: CHEMBL613223
ChEMBL Target Name: Mycolicibacter terrae
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard UnitsActivity Comment
MIC=0.1ug.mL-1
MICNot Determined
MIC=0.3ug.mL-1
MIC=0.7ug.mL-1
MICNot Determined
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Mycobacterium tuberculosis
External ID: CHEMBL3377975
Protocol: N/A
Comment: Journal: Bioorg Med Chem Lett
Year: 2014
Volume: 24
Issue: 14
First Page: 3118
Last Page: 3120
DOI: 10.1016/j.bmcl.2014.05.006

Target ChEMBL ID: CHEMBL360
ChEMBL Target Name: Mycobacterium tuberculosis
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
MIC=0.1ug.mL-1
MIC=12.5ug.mL-1
MIC=0.7ug.mL-1
MIC=1.5ug.mL-1
MIC=12.5ug.mL-1