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1879-77-2 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源：ChEMBL 靶标：Mineralocorticoid receptor
External ID: CHEMBL728550
Protocol: N/A
Comment: Journal: J Med Chem
Year: 1988
Volume: 31
Issue: 6
First Page: 1160
Last Page: 1169
DOI: 10.1021/jm00401a015

Target ChEMBL ID: CHEMBL3507
ChEMBL Target Name: Mineralocorticoid receptor
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: H - Homologous protein target assigned
Confidence: Homologous single protein target assigned
Standard TypeStandard RelationStandard Value
RBA=100
RBA=22
RBA=17
RBA=0.5
RBA=11
RBA=18
RBA=0.2
RBA=2.5
RBA=4.8
RBA=28
RBA=141
RBA=8
RBA=4
RBA=21
RBA=17
RBA<0.1
RBA=2.3
RBA=1.1
RBA=10
RBA=0.4
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源：ChEMBL 靶标：Glucocorticoid receptor
External ID: CHEMBL686331
Protocol: N/A
Comment: Journal: J Med Chem
Year: 1988
Volume: 31
Issue: 6
First Page: 1160
Last Page: 1169
DOI: 10.1021/jm00401a015

Target ChEMBL ID: CHEMBL3368
ChEMBL Target Name: Glucocorticoid receptor
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: H - Homologous protein target assigned
Confidence: Homologous single protein target assigned
Standard TypeStandard RelationStandard Value
RBA=9
RBA=2
RBA=80
RBA=0.2
RBA=8
RBA=55
RBA=5
RBA=9
RBA=38
RBA=4
RBA=40
RBA=260
RBA=0.3
RBA=100
RBA=15
RBA=300
RBA=37
RBA=47
RBA=30
RBA=18
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源：ChEMBL 靶标：Glucocorticoid receptor
External ID: CHEMBL686333
Protocol: N/A
Comment: Journal: J Med Chem
Year: 1988
Volume: 31
Issue: 6
First Page: 1160
Last Page: 1169
DOI: 10.1021/jm00401a015

Target ChEMBL ID: CHEMBL3368
ChEMBL Target Name: Glucocorticoid receptor
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: H - Homologous protein target assigned
Confidence: Homologous single protein target assigned
Standard TypeStandard RelationStandard Value
RBA=0.1
RBA<0.1
RBA=77
RBA=0.2
RBA=1.3
RBA=0.2
RBA=3
RBA=3.6
RBA=86
RBA<0.1
RBA=0.1
RBA=139
RBA<0.1
RBA=100
RBA=5
RBA=173
RBA=45
RBA=18
RBA=61
RBA=0.1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源：ChEMBL 靶标：Glucocorticoid receptor
External ID: CHEMBL686332
Protocol: N/A
Comment: Journal: J Med Chem
Year: 1988
Volume: 31
Issue: 6
First Page: 1160
Last Page: 1169
DOI: 10.1021/jm00401a015

Target ChEMBL ID: CHEMBL3368
ChEMBL Target Name: Glucocorticoid receptor
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: H - Homologous protein target assigned
Confidence: Homologous single protein target assigned
Standard TypeStandard RelationStandard Value
RBA=14
RBA=12
RBA=99
RBA=0.8
RBA=9
RBA=85
RBA=24
RBA=54
RBA=12
RBA=77
RBA=190
RBA=0.8
RBA=100
RBA=32
RBA=82
RBA=90
RBA=23
RBA=30
RBA=92
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源：ChEMBL 靶标：Progesterone receptor
External ID: CHEMBL763130
Protocol: N/A
Comment: Journal: J Med Chem
Year: 1988
Volume: 31
Issue: 6
First Page: 1160
Last Page: 1169
DOI: 10.1021/jm00401a015

Target ChEMBL ID: CHEMBL208
ChEMBL Target Name: Progesterone receptor
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: H - Homologous protein target assigned
Confidence: Homologous single protein target assigned
Standard TypeStandard RelationStandard Value
RBA=0.7
RBA=100
RBA=0.1
RBA=0.9
RBA<0.1
RBA=2.8
RBA=265
RBA=533
RBA<0.1
RBA=0.4
RBA=18
RBA=12
RBA=1.1
RBA=0.1
RBA<0.1
RBA=530
RBA<0.1
RBA=48
RBA<0.1
RBA=62
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源：ChEMBL 靶标：Glucocorticoid receptor
External ID: CHEMBL813557
Protocol: N/A
Comment: Journal: J Med Chem
Year: 1988
Volume: 31
Issue: 6
First Page: 1160
Last Page: 1169
DOI: 10.1021/jm00401a015

Target ChEMBL ID: CHEMBL3368
ChEMBL Target Name: Glucocorticoid receptor
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: H - Homologous protein target assigned
Confidence: Homologous single protein target assigned
Standard TypeStandard RelationStandard ValueStandard Units
Relative activity=49%
Relative activity=6%
Relative activity=106%
Relative activity=6%
Relative activity=91%
Relative activity=71%
Relative activity=6%
Relative activity=81%
Relative activity=11%
Relative activity=17%
Relative activity=127%
Relative activity=8%
Relative activity=100%
Relative activity=66%
Relative activity=98%
Relative activity=3%
Relative activity=99%
Relative activity=3.5%
Relative activity=45%
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源：ChEMBL 靶标：Glucocorticoid receptor
External ID: CHEMBL878587
Protocol: N/A
Comment: Journal: J Med Chem
Year: 1988
Volume: 31
Issue: 6
First Page: 1160
Last Page: 1169
DOI: 10.1021/jm00401a015

Target ChEMBL ID: CHEMBL3368
ChEMBL Target Name: Glucocorticoid receptor
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: H - Homologous protein target assigned
Confidence: Homologous single protein target assigned
Standard TypeStandard RelationStandard Value
RBA=8
RBA=17
RBA=84
RBA=0.3
RBA=3.3
RBA=22
RBA=1.2
RBA=6.5
RBA=63
RBA=3.3
RBA=24
RBA=174
RBA=0.4
RBA=100
RBA=13
RBA=300
RBA=33
RBA=33
RBA=34
RBA=12
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源：ChEMBL 靶标：Homo sapiens
External ID: CHEMBL700110
Protocol: N/A
Comment: Journal: J Med Chem
Year: 1986
Volume: 29
Issue: 11
First Page: 2125
Last Page: 2136
DOI: 10.1021/jm00161a001

Target ChEMBL ID: CHEMBL372
ChEMBL Target Name: Homo sapiens
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeActivity Comment
ActivityPotent
ActivityPotent
ActivityPotent
ActivityPotent
ActivityActive
ActivityPotent
ActivityActive
ActivityPotent
ActivityPotent
ActivityPotent
ActivityPotent
ActivityPotent
ActivityPotent
ActivityPotent
ActivityPotent
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源：ChEMBL 靶标：Androgen receptor
External ID: CHEMBL652299
Protocol: N/A
Comment: Journal: J Med Chem
Year: 1988
Volume: 31
Issue: 6
First Page: 1160
Last Page: 1169
DOI: 10.1021/jm00401a015

Target ChEMBL ID: CHEMBL3072
ChEMBL Target Name: Androgen Receptor
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: H - Homologous protein target assigned
Confidence: Homologous single protein target assigned
Standard TypeStandard RelationStandard Value
RBA=0.1
RBA=5.5
RBA=0.1
RBA=7.9
RBA<0.1
RBA=0.5
RBA=45
RBA=1.4
RBA<0.1
RBA=0.3
RBA=2.4
RBA=0.1
RBA=100
RBA=0.1
RBA<0.1
RBA=25
RBA<0.1
RBA=84
RBA<0.1
RBA=1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源：ChEMBL 靶标：Glucocorticoid receptor
External ID: CHEMBL686334
Protocol: N/A
Comment: Journal: J Med Chem
Year: 1988
Volume: 31
Issue: 6
First Page: 1160
Last Page: 1169
DOI: 10.1021/jm00401a015

Target ChEMBL ID: CHEMBL3368
ChEMBL Target Name: Glucocorticoid receptor
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: H - Homologous protein target assigned
Confidence: Homologous single protein target assigned
Standard TypeStandard RelationStandard Value
RBA=1.5
RBA=0.2
RBA=92
RBA=0.6
RBA=10
RBA=23
RBA=2.8
RBA=14
RBA=84
RBA<0.1
RBA=0.6
RBA=102
RBA=0.2
RBA=100
RBA=41
RBA=106
RBA=70
RBA=77
RBA=43
RBA=0.5
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源：ChEMBL 靶标：Glucocorticoid receptor
External ID: CHEMBL686335
Protocol: N/A
Comment: Journal: J Med Chem
Year: 1988
Volume: 31
Issue: 6
First Page: 1160
Last Page: 1169
DOI: 10.1021/jm00401a015

Target ChEMBL ID: CHEMBL3368
ChEMBL Target Name: Glucocorticoid receptor
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: H - Homologous protein target assigned
Confidence: Homologous single protein target assigned
Standard TypeStandard RelationStandard Value
RBA=14
RBA=42
RBA=92
RBA=1.1
RBA=3.4
RBA=67
RBA=22
RBA=75
RBA=9.3
RBA=50
RBA=141
RBA=0.9
RBA=100
RBA=31
RBA=280
RBA=58
RBA=96
RBA=16
RBA=22
RBA=67

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