HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Receptor-type tyrosine-protein kinase FLT3

External ID: CHEMBL3794752

Protocol: N/A

Comment: Compounds with activity <= 10uM or explicitly reported as active by ChEMBL are flagged as active in this PubChem assay presentation.

Journal: Bioorg. Med. Chem. Lett.
Year: 2016
Volume: 26
Issue: 9
First Page: 2370
Last Page: 2374
DOI: 10.1016/j.bmcl.2016.03.006

Target ChEMBL ID: CHEMBL1974
ChEMBL Target Name: Tyrosine-protein kinase receptor FLT3
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

PubChem Standard Value	Standard Type	Standard Relation	Standard Value	Standard Units
0.061	IC50	=	61	nM
0.046	IC50	=	46	nM
0.042	IC50	=	42	nM
2	IC50	>	2000	nM
0.552	IC50	=	552	nM
0.443	IC50	=	443	nM
2	IC50	>	2000	nM
0.107	IC50	=	107	nM
2	IC50	>	2000	nM

17954-06-2 靶点实验数据