HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Mus musculus

External ID: CHEMBL4734818

Protocol: N/A

Comment: Journal: Eur J Med Chem
Year: 2021
Volume: 213
First Page: 113042
Last Page: 113042
DOI: 10.1016/j.ejmech.2020.113042

Target ChEMBL ID: CHEMBL375
ChEMBL Target Name: Mus musculus
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular

Standard Type	Activity Comment
Activity	Not Active

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：N/A

External ID: CHEMBL4734851

Protocol: N/A

Comment: Journal: Eur J Med Chem
Year: 2021
Volume: 213
First Page: 113042
Last Page: 113042
DOI: 10.1016/j.ejmech.2020.113042

Standard Type	Activity Comment
Activity	Toxic
Activity	Non-Toxic
Activity	Non-Toxic
Activity	Non-Toxic
Activity	Non-Toxic

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Mus musculus

External ID: CHEMBL4734819

Protocol: N/A

Comment: Journal: Eur J Med Chem
Year: 2021
Volume: 213
First Page: 113042
Last Page: 113042
DOI: 10.1016/j.ejmech.2020.113042

Target ChEMBL ID: CHEMBL375
ChEMBL Target Name: Mus musculus
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular

Standard Type	Activity Comment
Activity	Not Active

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：N/A

External ID: CHEMBL4734816

Protocol: N/A

Comment: Journal: Eur J Med Chem
Year: 2021
Volume: 213
First Page: 113042
Last Page: 113042
DOI: 10.1016/j.ejmech.2020.113042

Standard Type	Activity Comment
Activity	Non-Toxic

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：N/A

External ID: CHEMBL4734849

Protocol: N/A

Comment: Journal: Eur J Med Chem
Year: 2021
Volume: 213
First Page: 113042
Last Page: 113042
DOI: 10.1016/j.ejmech.2020.113042

Standard Type	Activity Comment
Activity	Toxic
Activity	Non-Toxic
Activity	Non-Toxic
Activity	Non-Toxic
Activity	Non-Toxic

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：N/A

External ID: CHEMBL4734810

Protocol: N/A

Comment: Journal: Eur J Med Chem
Year: 2021
Volume: 213
First Page: 113042
Last Page: 113042
DOI: 10.1016/j.ejmech.2020.113042

Standard Type	Standard Relation	Standard Value	Standard Units
Drug metabolism	=	1731	pmol
Drug metabolism	=	1002	pmol
Drug metabolism	=	82	pmol
Drug metabolism	=	283	pmol
Drug metabolism	=	58	pmol

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Mus musculus

External ID: CHEMBL4734814

Protocol: N/A

Comment: Journal: Eur J Med Chem
Year: 2021
Volume: 213
First Page: 113042
Last Page: 113042
DOI: 10.1016/j.ejmech.2020.113042

Target ChEMBL ID: CHEMBL375
ChEMBL Target Name: Mus musculus
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular

Standard Type	Activity Comment
Activity	Dose-dependent effect
Activity	Dose-dependent effect

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Mus musculus

External ID: CHEMBL4734815

Protocol: N/A

Comment: Journal: Eur J Med Chem
Year: 2021
Volume: 213
First Page: 113042
Last Page: 113042
DOI: 10.1016/j.ejmech.2020.113042

Target ChEMBL ID: CHEMBL375
ChEMBL Target Name: Mus musculus
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular

Standard Type	Activity Comment
Activity	Dose-dependent effect
Activity	Dose-dependent effect

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：N/A

External ID: CHEMBL4734812

Protocol: N/A

Comment: Journal: Eur J Med Chem
Year: 2021
Volume: 213
First Page: 113042
Last Page: 113042
DOI: 10.1016/j.ejmech.2020.113042

Standard Type	Standard Relation	Standard Value	Standard Units
Drug metabolism	=	161	pmol
Drug metabolism	=	24	pmol
Drug metabolism	=	190	pmol
Drug metabolism	=	42	pmol
Drug metabolism	=	58	pmol

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Fatty-acid amide hydrolase 1

External ID: CHEMBL4734806

Protocol: N/A

Comment: Journal: Eur J Med Chem
Year: 2021
Volume: 213
First Page: 113042
Last Page: 113042
DOI: 10.1016/j.ejmech.2020.113042

Target ChEMBL ID: CHEMBL3455
ChEMBL Target Name: Anandamide amidohydrolase
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

Standard Type	Standard Relation	Standard Value	Standard Units
Drug metabolism	=	12	nmol
Drug metabolism	=	8.8	nmol
Drug metabolism	=	0.54	nmol
Drug metabolism	=	2.5	nmol
Drug metabolism	=	3	nmol
Drug metabolism	=	2.5	nmol

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：N/A

External ID: CHEMBL4734807

Protocol: N/A

Comment: Journal: Eur J Med Chem
Year: 2021
Volume: 213
First Page: 113042
Last Page: 113042
DOI: 10.1016/j.ejmech.2020.113042

Standard Type	Standard Relation	Standard Value	Standard Units
Drug metabolism	=	0.09	nmol
Drug metabolism	=	0.05	nmol
Drug metabolism	=	0.005	nmol
Drug metabolism	=	0.01	nmol
Drug metabolism	=	0.06	nmol
Drug metabolism	=	0.04	nmol

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Mus musculus

External ID: CHEMBL4734824

Protocol: N/A

Comment: Journal: Eur J Med Chem
Year: 2021
Volume: 213
First Page: 113042
Last Page: 113042
DOI: 10.1016/j.ejmech.2020.113042

Target ChEMBL ID: CHEMBL375
ChEMBL Target Name: Mus musculus
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular

Standard Type	Activity Comment
Activity	Active

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Mus musculus

External ID: CHEMBL4734825

Protocol: N/A

Comment: Journal: Eur J Med Chem
Year: 2021
Volume: 213
First Page: 113042
Last Page: 113042
DOI: 10.1016/j.ejmech.2020.113042

Target ChEMBL ID: CHEMBL375
ChEMBL Target Name: Mus musculus
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular

Standard Type	Activity Comment
Activity	Active

1687-53-2 靶点实验数据