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1621908-92-6 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:BindingDB 靶标:N/A
External ID: BindingDB_590_1
Protocol: N/A
Comment: Compounds with any of Ki, IC50, Kd, or EC50 activity value <= 10uM are labeled as "Active".
If multiple measurements are available for a given compound, it is labeled as "Active" if any of the measurements meet the criterion. Activity values are checked in the order of Ki, IC50, Kd, and EC50. The first entry that meets the above activity threshold is used to determine "Standard Type", "Standard Relation", and "PubChem Standard Value". Otherwise, the first non-empty entry will be used to set those values.
Standard TypePubChem Standard ValueEC50Target Accession(s)LigandTarget
EC500.33330P08173BDBM280373Muscarinic acetylcholine receptor M4
EC502.262260P08173BDBM280401Muscarinic acetylcholine receptor M4
EC500.18180P08173BDBM280403Muscarinic acetylcholine receptor M4
EC500.0990P08173BDBM280404Muscarinic acetylcholine receptor M4
EC506.736730P08173BDBM280406Muscarinic acetylcholine receptor M4
EC500.0330P08173BDBM280408Muscarinic acetylcholine receptor M4
EC500.74740P08173BDBM280409Muscarinic acetylcholine receptor M4
EC500.25250P08173BDBM280418Muscarinic acetylcholine receptor M4
EC500.21210P08173BDBM280419Muscarinic acetylcholine receptor M4
EC500.12120P08173BDBM280436Muscarinic acetylcholine receptor M4
EC500.21210P08173BDBM280440Muscarinic acetylcholine receptor M4
EC501.051050P08173BDBM280444Muscarinic acetylcholine receptor M4
EC500.85850P08173BDBM280450Muscarinic acetylcholine receptor M4
EC500.08585P08173BDBM280451Muscarinic acetylcholine receptor M4