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1443237-36-2 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:BindingDB 靶标:N/A
External ID: BindingDB_6824_1
Protocol: N/A
Comment: Compounds with any of Ki, IC50, Kd, or EC50 activity value <= 10uM are labeled as "Active".
If multiple measurements are available for a given compound, it is labeled as "Active" if any of the measurements meet the criterion. Activity values are checked in the order of Ki, IC50, Kd, and EC50. The first entry that meets the above activity threshold is used to determine "Standard Type", "Standard Relation", and "PubChem Standard Value". Otherwise, the first non-empty entry will be used to set those values.
Standard TypeStandard RelationPubChem Standard ValueIC50 QualifierIC50Target Accession(s)LigandTarget
IC500.273273O60674BDBM153130Tyrosine-protein kinase JAK2
IC500.00575.7P52333BDBM153131Tyrosine-protein kinase JAK3
IC500.07373O60674BDBM153132Tyrosine-protein kinase JAK2
IC500.00464.6P52333BDBM153133Tyrosine-protein kinase JAK3
IC500.06262O60674BDBM153134Tyrosine-protein kinase JAK2
IC500.00757.5P52333BDBM153135Tyrosine-protein kinase JAK3
IC500.125125O60674BDBM153135Tyrosine-protein kinase JAK2
IC500.00818.1P52333BDBM153136Tyrosine-protein kinase JAK3
IC500.339339O60674BDBM153136Tyrosine-protein kinase JAK2
IC500.00464.6P52333BDBM153137Tyrosine-protein kinase JAK3
IC500.215215O60674BDBM153138Tyrosine-protein kinase JAK2
IC500.00575.7P52333BDBM153139Tyrosine-protein kinase JAK3
IC500.145145O60674BDBM153140Tyrosine-protein kinase JAK2
IC500.00888.8P52333BDBM153141Tyrosine-protein kinase JAK3
IC500.186186O60674BDBM153141Tyrosine-protein kinase JAK2
IC500.00757.5P52333BDBM153142Tyrosine-protein kinase JAK3
IC500.168168O60674BDBM153142Tyrosine-protein kinase JAK2
IC500.0099P52333BDBM153143Tyrosine-protein kinase JAK3
IC500.121121O60674BDBM153143Tyrosine-protein kinase JAK2
IC500.00424.2P52333BDBM153144Tyrosine-protein kinase JAK3