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142-78-9 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL872905
Protocol: N/A
Comment: Journal: Bioorg Med Chem Lett
Year: 2007
Volume: 17
Issue: 11
First Page: 3231
Last Page: 3234
DOI: 10.1016/j.bmcl.2007.03.013
Standard TypeStandard RelationStandard ValueStandard Units
Solubility=0.34g
Solubility=9.14g
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL4420713
Protocol: N/A
Comment: Data Source: SureChEMBL Patent Bioactivity Data
Standard TypeStandard RelationStandard ValueStandard Units
Inhibition=35%
Inhibition=11%
Inhibition=22%
Inhibition=59%
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL872903
Protocol: N/A
Comment: Journal: Bioorg Med Chem Lett
Year: 2007
Volume: 17
Issue: 11
First Page: 3231
Last Page: 3234
DOI: 10.1016/j.bmcl.2007.03.013
Standard TypeStandard RelationStandard ValueStandard Units
Solubility=0.16g
Solubility=1.76g
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Diacylglycerol O-acyltransferase 1
External ID: CHEMBL4420716
Protocol: N/A
Comment: Target ChEMBL ID: CHEMBL4523395
ChEMBL Target Name: Diacylglycerol O-acyltransferase 1
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

Data Source: SureChEMBL Patent Bioactivity Data
Standard TypeStandard RelationStandard ValueStandard Units
Inhibition=12%
Inhibition=32%
Inhibition=28%
Inhibition=23%
Inhibition=64%
Inhibition=21%
Inhibition=35%
Inhibition=30%
Inhibition=13%
Inhibition=34%
Inhibition=81%
Inhibition=45%
Inhibition=20%
Inhibition=25%
Inhibition=12%
Inhibition=33%
Inhibition=26%
Inhibition=20%
Inhibition=20%
Inhibition=76%
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL872904
Protocol: N/A
Comment: Journal: Bioorg Med Chem Lett
Year: 2007
Volume: 17
Issue: 11
First Page: 3231
Last Page: 3234
DOI: 10.1016/j.bmcl.2007.03.013
Standard TypeStandard RelationStandard ValueStandard Units
Solubility=0.03g
Solubility=0.38g
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Lecithin retinol acyltransferase
External ID: CHEMBL4420718
Protocol: N/A
Comment: Target ChEMBL ID: CHEMBL4523439
ChEMBL Target Name: Lecithin retinol acyltransferase
ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain
Relationship Type: D - Direct protein target assigned
Confidence: Direct single protein target assigned

Data Source: SureChEMBL Patent Bioactivity Data
Standard TypeStandard RelationStandard ValueStandard Units
Inhibition=0%
Inhibition=0%
Inhibition=33%
Inhibition=43%
Inhibition=28%
Inhibition=35%
Inhibition=0%
Inhibition=34%
Inhibition=15%
Inhibition=77%
Inhibition=49%
Inhibition=4%
Inhibition=14%
Inhibition=25%
Inhibition=71%
Inhibition=38%
Inhibition=33%
Inhibition=36%
Inhibition=79%
Inhibition=16%