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117983-41-2 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL630220
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1989
Volume: 32
Issue: 2
First Page: 504
Last Page: 516
DOI: 10.1021/jm00122a035
Standard TypeStandard RelationStandard Value
LogD=-0.45
LogD=-0.36
LogD=-1.3
LogD=-0.87
LogD=-1.71
LogD=-1.41
LogD=-0.47
LogD=-1.4
LogD=-0.7
LogD=-1.55
LogD=-2.1
LogD=-1.49
LogD=-1.74
LogD=-1.4
LogD=-2.36
LogD=-1.1
LogD=-1.99
LogD=-1.62
LogD=-2.14
LogD=0.31
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Mus musculus
External ID: CHEMBL739615
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1989
Volume: 32
Issue: 2
First Page: 504
Last Page: 516
DOI: 10.1021/jm00122a035

Target ChEMBL ID: CHEMBL375
ChEMBL Target Name: Mus musculus
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard Value
Survival=2
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Mus musculus
External ID: CHEMBL739704
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1989
Volume: 32
Issue: 2
First Page: 504
Last Page: 516
DOI: 10.1021/jm00122a035

Target ChEMBL ID: CHEMBL375
ChEMBL Target Name: Mus musculus
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard ValueStandard Units
LD50=850umol.kg-1
LD50=860umol.kg-1
LD50=4500umol.kg-1
LD50=860umol.kg-1
LD50=650umol.kg-1
LD50=390umol.kg-1
LD50=600umol.kg-1
LD50=430umol.kg-1
LD50=310umol.kg-1
LD50=430umol.kg-1
LD50=150umol.kg-1
LD50=270umol.kg-1
LD50=420umol.kg-1
LD50=430umol.kg-1
LD50=510umol.kg-1
LD50=640umol.kg-1
LD50=620umol.kg-1
LD50=330umol.kg-1
LD50=910umol.kg-1
LD50=440umol.kg-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Mus musculus
External ID: CHEMBL879316
Protocol: N/A
Comment: Journal: J Med Chem
Year: 1989
Volume: 32
Issue: 2
First Page: 504
Last Page: 516
DOI: 10.1021/jm00122a035

Target ChEMBL ID: CHEMBL375
ChEMBL Target Name: Mus musculus
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard Value
Survival=0
Survival=0
Survival=10
Survival=1
Survival=0
Survival=0
Survival=1
Survival=2
Survival=0
Survival=0
Survival=3
Survival=
Survival=4
Survival=1
Survival=0
Survival=3
Survival=9
Survival=1
Survival=0
Survival=6
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:Mus musculus
External ID: CHEMBL739614
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1989
Volume: 32
Issue: 2
First Page: 504
Last Page: 516
DOI: 10.1021/jm00122a035

Target ChEMBL ID: CHEMBL375
ChEMBL Target Name: Mus musculus
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular
Standard TypeStandard RelationStandard Value
Survival=0
Survival=0
Survival=9
Survival=0
Survival=0
Survival=0
Survival=0
Survival=0
Survival=0
Survival=1
Survival=3
Survival=3
Survival=0
Survival=4
Survival=4
Survival=0
Survival=0
Survival=4
Survival=1
Survival=1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL632263
Protocol: N/A
Comment: Journal: J. Med. Chem.
Year: 1989
Volume: 32
Issue: 2
First Page: 504
Last Page: 516
DOI: 10.1021/jm00122a035
Standard TypeStandard RelationStandard Value
pKa=8.05
pKa=8.11
pKa=7.94
pKa=7.99
pKa=8.23
pKa=8.03
pKa=8.04
pKa=8
pKa=8
pKa=8.2
pKa=7.99
pKa=8.03
pKa=8.06
pKa=7.99
pKa=8.02
pKa=8.04
pKa=7.98
pKa=7.96
pKa=8.06
pKa=8.18