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1069-29-0 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL4427183
Protocol: N/A
Comment: Journal: J Med Chem
Year: 2016
Volume: 59
Issue: 15
First Page: 7293
Last Page: 7298
DOI: 10.1021/acs.jmedchem.6b00647
Standard TypeStandard UnitsActivity Comment
Inhibition%Active
Inhibition%Active
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL4427184
Protocol: N/A
Comment: Journal: J Med Chem
Year: 2016
Volume: 59
Issue: 15
First Page: 7293
Last Page: 7298
DOI: 10.1021/acs.jmedchem.6b00647
Standard TypeStandard UnitsActivity Comment
Inhibition%Active
Inhibition%Active
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL4427175
Protocol: N/A
Comment: Journal: J Med Chem
Year: 2016
Volume: 59
Issue: 15
First Page: 7293
Last Page: 7298
DOI: 10.1021/acs.jmedchem.6b00647
Standard TypeStandard RelationStandard Value
Ratio=0.21
Ratio=0.3
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL4427176
Protocol: N/A
Comment: Journal: J Med Chem
Year: 2016
Volume: 59
Issue: 15
First Page: 7293
Last Page: 7298
DOI: 10.1021/acs.jmedchem.6b00647
Standard TypeStandard RelationStandard Value
Ratio=0.27
Ratio=0.32
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL4427177
Protocol: N/A
Comment: Journal: J Med Chem
Year: 2016
Volume: 59
Issue: 15
First Page: 7293
Last Page: 7298
DOI: 10.1021/acs.jmedchem.6b00647
Standard TypeStandard RelationStandard Value
Ratio=0.4
Ratio=0.52
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL4427178
Protocol: N/A
Comment: Journal: J Med Chem
Year: 2016
Volume: 59
Issue: 15
First Page: 7293
Last Page: 7298
DOI: 10.1021/acs.jmedchem.6b00647
Standard TypeStandard RelationStandard ValueStandard Units
T1/2=2.64hr
T1/2=475.2hr