HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Mycobacterium tuberculosis

External ID: CHEMBL925897

Protocol: N/A

Comment: Journal: J. Nat. Prod.
Year: 2008
Volume: 71
Issue: 3
First Page: 438
Last Page: 444
DOI: 10.1021/np700738k

Target ChEMBL ID: CHEMBL360
ChEMBL Target Name: Mycobacterium tuberculosis
ChEMBL Target Type: ORGANISM - Target is a complete organism
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular

Standard Type	Standard Relation	Standard Value	Standard Units
Activity	=	99	%
MIC	=	6.25	ug.mL-1

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：MCF7

External ID: CHEMBL925906

Protocol: N/A

Comment: Journal: J. Nat. Prod.
Year: 2008
Volume: 71
Issue: 3
First Page: 438
Last Page: 444
DOI: 10.1021/np700738k

Target ChEMBL ID: CHEMBL387
ChEMBL Target Name: MCF7
ChEMBL Target Type: CELL-LINE - Target is a specific cell-line
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular

Standard Type	Standard Relation	Standard Value	Standard Units
Activity	=	2.5	ug ml-1
Activity	=	5.1	ug ml-1
Activity	=	0.047	ug ml-1
Activity	=	0.41	ug ml-1

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：SF-268

External ID: CHEMBL925907

Protocol: N/A

Comment: Journal: J. Nat. Prod.
Year: 2008
Volume: 71
Issue: 3
First Page: 438
Last Page: 444
DOI: 10.1021/np700738k

Target ChEMBL ID: CHEMBL613977
ChEMBL Target Name: SF-268
ChEMBL Target Type: CELL-LINE - Target is a specific cell-line
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular

Standard Type	Standard Relation	Standard Value	Standard Units
Activity	=	1.7	ug ml-1
Activity	=	4.4	ug ml-1
Activity	=	0.21	ug ml-1
Activity	=	0.42	ug ml-1

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：DU-145

External ID: CHEMBL925909

Protocol: N/A

Comment: Journal: J. Nat. Prod.
Year: 2008
Volume: 71
Issue: 3
First Page: 438
Last Page: 444
DOI: 10.1021/np700738k

Target ChEMBL ID: CHEMBL613508
ChEMBL Target Name: DU-145
ChEMBL Target Type: CELL-LINE - Target is a specific cell-line
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular

Standard Type	Standard Relation	Standard Value	Standard Units
Activity	=	1.9	ug ml-1
Activity	=	7.3	ug ml-1
Activity	=	0.13	ug ml-1
Activity	=	0.0017	ug ml-1
Activity	=	0.0021	ug ml-1
Activity	=	0.27	ug ml-1
Activity	=	0.0098	ug ml-1
Activity	>	1	ug ml-1
Activity	=	0.6	ug ml-1
Activity	=	0.0056	ug ml-1

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：NCI-H460

External ID: CHEMBL925902

Protocol: N/A

Comment: Journal: J. Nat. Prod.
Year: 2008
Volume: 71
Issue: 3
First Page: 438
Last Page: 444
DOI: 10.1021/np700738k

Target ChEMBL ID: CHEMBL396
ChEMBL Target Name: NCI-H460
ChEMBL Target Type: CELL-LINE - Target is a specific cell-line
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular

Standard Type	Standard Relation	Standard Value	Standard Units
Activity	=	1.5	ug ml-1
Activity	>	10	ug ml-1
Activity	=	0.28	ug ml-1
Activity	=	0.0018	ug ml-1
Activity	=	7.7E-4	ug ml-1
Activity	=	0.21	ug ml-1
Activity	=	0.022	ug ml-1
Activity	=	0.28	ug ml-1
Activity	=	0.36	ug ml-1
Activity	=	5.4E-4	ug ml-1

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：MDCK

External ID: CHEMBL1066303

Protocol: N/A

Comment: Journal: J. Med. Chem.
Year: 2010
Volume: 53
Issue: 1
First Page: 61
Last Page: 76
DOI: 10.1021/jm900672t

Target ChEMBL ID: CHEMBL614068
ChEMBL Target Name: MDCK
ChEMBL Target Type: CELL-LINE - Target is a specific cell-line
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular

Standard Type	Standard Relation	Standard Value	Standard Units
Papp	=	17	10'-6 cm/s
Papp	=	1.9	10'-6 cm/s
Papp	=	0.87	10'-6 cm/s

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：KM-20L2

External ID: CHEMBL925903

Protocol: N/A

Comment: Journal: J. Nat. Prod.
Year: 2008
Volume: 71
Issue: 3
First Page: 438
Last Page: 444
DOI: 10.1021/np700738k

Target ChEMBL ID: CHEMBL614791
ChEMBL Target Name: KM-20L2
ChEMBL Target Type: CELL-LINE - Target is a specific cell-line
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular

Standard Type	Standard Relation	Standard Value	Standard Units
Activity	=	3.7	ug ml-1
Activity	=	8.8	ug ml-1
Activity	=	0.022	ug ml-1
Activity	=	0.0014	ug ml-1
Activity	=	0.0076	ug ml-1
Activity	=	0.19	ug ml-1
Activity	=	0.022	ug ml-1
Activity	>	1	ug ml-1
Activity	=	0.37	ug ml-1
Activity	=	0.0049	ug ml-1

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：BXPC-3

External ID: CHEMBL925905

Protocol: N/A

Comment: Journal: J. Nat. Prod.
Year: 2008
Volume: 71
Issue: 3
First Page: 438
Last Page: 444
DOI: 10.1021/np700738k

Target ChEMBL ID: CHEMBL614530
ChEMBL Target Name: BXPC-3
ChEMBL Target Type: CELL-LINE - Target is a specific cell-line
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular

Standard Type	Standard Relation	Standard Value	Standard Units
Activity	=	2.5	ug ml-1
Activity	=	6.2	ug ml-1
Activity	=	0.07	ug ml-1
Activity	=	4.4E-4	ug ml-1
Activity	=	0.0012	ug ml-1
Activity	=	0.25	ug ml-1
Activity	=	0.024	ug ml-1
Activity	>	1	ug ml-1
Activity	=	0.35	ug ml-1
Activity	=	0.027	ug ml-1

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：Vero

External ID: CHEMBL925898

Protocol: N/A

Comment: Journal: J. Nat. Prod.
Year: 2008
Volume: 71
Issue: 3
First Page: 438
Last Page: 444
DOI: 10.1021/np700738k

Target ChEMBL ID: CHEMBL391
ChEMBL Target Name: Vero
ChEMBL Target Type: CELL-LINE - Target is a specific cell-line
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular

Standard Type	Standard Relation	Standard Value	Standard Units
IC50	=	1.7	ug.mL-1

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16

来源：ChEMBL 靶标：P388

External ID: CHEMBL925899

Protocol: N/A

Comment: Journal: J. Nat. Prod.
Year: 2008
Volume: 71
Issue: 3
First Page: 438
Last Page: 444
DOI: 10.1021/np700738k

Target ChEMBL ID: CHEMBL389
ChEMBL Target Name: P388
ChEMBL Target Type: CELL-LINE - Target is a specific cell-line
Relationship Type: N - Non-molecular target assigned
Confidence: Target assigned is non-molecular

Standard Type	Standard Relation	Standard Value	Standard Units
Activity	=	0.23	ug ml-1
Activity	=	0.029	ug ml-1
Activity	=	0.0031	ug ml-1
Activity	=	0.0023	ug ml-1
Activity	>	1	ug ml-1
Activity	=	2.4	ug ml-1
Activity	=	0.21	ug ml-1
Activity	=	0.0027	ug ml-1
Activity	=	0.21	ug ml-1
Activity	=	5	ug ml-1
Activity	=	0.0067	ug ml-1
Activity	=	0.008	ug ml-1
Activity	=	0.12	ug ml-1
Activity	=	0.037	ug ml-1
Activity	<	0.001	ug ml-1

104264-80-4 靶点实验数据