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1032902-80-9 靶点实验数据

HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL4716867
Protocol: N/A
Comment: Journal: Bioorg Med Chem Lett
Year: 2016
Volume: 26
Issue: 3.0
First Page: 1090
Last Page: 1096
DOI: 10.1016/j.bmcl.2015.11.049
Standard TypeStandard RelationStandard Value
log(permeability)=-4.1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL4716864
Protocol: N/A
Comment: Journal: Bioorg Med Chem Lett
Year: 2016
Volume: 26
Issue: 3.0
First Page: 1090
Last Page: 1096
DOI: 10.1016/j.bmcl.2015.11.049
Standard TypeStandard RelationStandard ValueStandard Units
CL=32mL.min-1.g-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL4716887
Protocol: N/A
Comment: Journal: Bioorg Med Chem Lett
Year: 2016
Volume: 26
Issue: 3.0
First Page: 1090
Last Page: 1096
DOI: 10.1016/j.bmcl.2015.11.049
Standard TypeStandard RelationStandard Value
Ratio IC50=20
Ratio IC50=20
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL4716868
Protocol: N/A
Comment: Journal: Bioorg Med Chem Lett
Year: 2016
Volume: 26
Issue: 3.0
First Page: 1090
Last Page: 1096
DOI: 10.1016/j.bmcl.2015.11.049
Standard TypeStandard RelationStandard ValueStandard Units
permeability=2.6cm/s
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL4716869
Protocol: N/A
Comment: Journal: Bioorg Med Chem Lett
Year: 2016
Volume: 26
Issue: 3.0
First Page: 1090
Last Page: 1096
DOI: 10.1016/j.bmcl.2015.11.049
Standard TypeStandard RelationStandard ValueStandard Units
permeability=3.1cm/s
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL4716862
Protocol: N/A
Comment: Journal: Bioorg Med Chem Lett
Year: 2016
Volume: 26
Issue: 3.0
First Page: 1090
Last Page: 1096
DOI: 10.1016/j.bmcl.2015.11.049
Standard TypeStandard RelationStandard ValueStandard Units
CL=37mL.min-1.g-1
HepG2 Cytotoxicity Assay Measured in Cell-Based System Using Plate Reader - 7071-02_Inhibitor_Dose_DryPowder_Activity_Set16
来源:ChEMBL 靶标:N/A
External ID: CHEMBL4716863
Protocol: N/A
Comment: Journal: Bioorg Med Chem Lett
Year: 2016
Volume: 26
Issue: 3.0
First Page: 1090
Last Page: 1096
DOI: 10.1016/j.bmcl.2015.11.049
Standard TypeStandard RelationStandard ValueStandard Units
CL=30mL.min-1.g-1