177702-21-5

• 常用中文名：(R)-1-boc-4-(氨基羧基甲基)哌啶
• 常用英文名：(R)-1-BOC-4-(AMINOCARBOXYMETHYL)PIPERIDINE
• CAS号：177702-21-5
• 分子式：C₁₂H₂₂N₂O₄
• 分子量：258.31400
• 发布时间：2018-12-17 09:06:09
• 更新时间：2025-08-25 11:40:20

名称

• 中文名: (R)-1-boc-4-(氨基羧基甲基)哌啶
• 英文名: (2R)-2-amino-2-[1-[(2-methylpropan-2-yl)oxycarbonyl]piperidin-4-yl]acetic acid
• 中文别名: (R)-2-氨基-2-(1-(叔丁氧羰基)哌啶-4-基)乙酸; (R)-1-BOC-4-(氨基羧甲基)哌啶; (R)-2-氨基-2-(1-Boc-4-哌啶基)乙酸; (R)-1-BOC-4-(氨基羧基甲基)哌啶
• 英文别名: (R)-4-(Amino-cboxy-methyl)-piperidine-1-cboxylic acid tert-butyl ester; (R)-a-Amino-1-Boc-4-piperidineacetic acid; (R)-2-Amino-2-(1-(tert-butoxycbonyl)piperidin-4-yl)acetic acid; (2R)-2-amino-2-[1-[(2-methylpropan-2-yl)oxycbonyl]piperidin-4-yl]acetic acid; 4-Piperidineacetic acid, α-amino-1-[(1,1-dimethylethoxy)carbonyl]-, (αR); (R)-2-Amino-2-(1-Boc-4-piperidyl)acetic Acid; 4-((R)-amino-cboxy-methyl)piperidine-1-cboxylic acid tert-butyl ester; (2R)-2-amino-2-(1-tert-butoxycbonyl-4-piperidyl)acetic acid; (R)-1-BOC-4-(AMINOCBOXYMETHYL)PIPERIDINE

物化性质

• 密度: 1.181g/cm3
• 沸点: 397.9ºC at 760 mmHg
• 分子式: C₁₂H₂₂N₂O₄
• 分子量: 258.31400
• 闪点: 194.5ºC
• 精确质量: 258.15800
• PSA: 92.86000
• LogP: 1.68360
• 蒸汽压: 1.92E-07mmHg at 25°C
• 折射率: 1.513

安全

• 海关编码: 2933399090

合成路线

400888-22-4 ~82% 177702-21-5

文献：Shieh, Wen-Chung; Xue, Song; Reel, Noela; Wu, Raeann; Fitt, John; Repic, Oljan Tetrahedron Asymmetry, 2001 , vol. 12, # 17 p. 2421 - 2425

161315-57-7 ~83% 177702-21-5

文献：Monovich, Lauren G.; Tommasi, Ruben A.; Fujimoto, Roger A.; Blancuzzi, Vincent; Clark, Kirk; Cornell, Wendy D.; Doti, Robert; Doughty, John; Fang, James; Farley, David; Fitt, John; Ganu, Vishwas; Goldberg, Ronald; Goldstein, Robert; Lavoie, Stacey; Kulathila, Raviraj; Macchia, William; Parker, David T.; Melton, Richard; O'Byrne, Elizabeth; Pastor, Gary; Pellas, Theodore; Quadros, Elizabeth; Reel, Noela; Roland, Dennis M.; Sakane, Yumi; Singh, Hem; Skiles, Jerry; Somers, Joseph; Toscano, Karen; Wigg, Andrew; Zhou, Siyuan; Zhu, Lijuan; Shieh, Wen-Chung; Xue, Song; McQuire, Leslie W. Journal of Medicinal Chemistry, 2009 , vol. 52, # 11 p. 3523 - 3538

79099-07-3 ~% 177702-21-5

文献：Shieh, Wen-Chung; Xue, Song; Reel, Noela; Wu, Raeann; Fitt, John; Repic, Oljan Tetrahedron Asymmetry, 2001 , vol. 12, # 17 p. 2421 - 2425

400888-21-3 ~% 177702-21-5

文献：Shieh, Wen-Chung; Xue, Song; Reel, Noela; Wu, Raeann; Fitt, John; Repic, Oljan Tetrahedron Asymmetry, 2001 , vol. 12, # 17 p. 2421 - 2425

313491-20-2 ~% 177702-21-5

文献：Shieh, Wen-Chung; Xue, Song; Reel, Noela; Wu, Raeann; Fitt, John; Repic, Oljan Tetrahedron Asymmetry, 2001 , vol. 12, # 17 p. 2421 - 2425

上下游产品

上游产品  3
400888-22-4 79099-07-3 313491-20-2
下游产品  0

海关

海关编码	2933399090
中文概述	2933399090. 其他结构含非稠合吡啶环的化合物. 增值税率:17.0%. 退税率:13.0%. 监管条件:无. 最惠国关税:6.5%. 普通关税:20.0%
申报要素	品名, 成分含量, 用途, 乌洛托品请注明外观, 6－己内酰胺请注明外观, 签约日期
Summary	2933399090. other compounds containing an unfused pyridine ring (whether or not hydrogenated) in the structure. VAT:17.0%. Tax rebate rate:13.0%. . MFN tariff:6.5%. General tariff:20.0%