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Dimerization of pyrazolyl??5??hydroxypyrrolidinones to tetrazocines

: Brinkmeyer, Raymond S.; Terando, Norman H. Journal of Heterocyclic Chemistry, 1989 , vol. 26, p. 1713 - 1717

Abstract The dimerization of the hydroxypyrrolidinones 5 and 9 yield the tetrazocines 8 and 11. In addition, in the case of compound 9, the ring-fused hexaazacyclododecane 12 was isolated. X-ray diffraction analysis of compound 11 verified the dimeric structu...

n??Butyllithium??mediated reactions of 1??(2??azidoarylmethyl)??1H??benzotriazoles with alkyl halides

: Journal of Heterocyclic Chemistry, , vol. 47, # 1 p. 98 - 111

... Journal of Heterocyclic Chemistry: Previous article in issue: Unusual anisotropic effects from 1,3-dipolar cycloadducts of 4 ... J. Heterocyclic Chem., 2010. ... of nitrene [3]. Nitrene is known as a useful reactive species for the synthesis of nitrogen-c...

Study of the reactivity of α??acylenaminoketones. Synthesis of pyrazoles

: Journal of Heterocyclic Chemistry, , vol. 38, # 1 p. 109 - 123

... J. Heterocyclic Chem., 38, 109 (2001). ... Amongst pyrazole derivatives, C-aminopyrazoles are the most used in heterocyclic chemistry as starting materials because of their ... of the different ways that the two ketonic carbonyls could react; different ki...

Die polonovski??reaktion an 3, 4??dihydro??4??methyl??2H??1, 4??benzoxazin??2??carbonsäurederivaten; ein neuer syntheseweg zu 4H??1, 4??benzoxazinen. 10. Mitteilung …

: Bartsch, Herbert; Schwarz, Otto Journal of Heterocyclic Chemistry, 1982 , vol. 19, p. 1189 - 1193

Abstract Die Dihydro-1, 4-benzoxazin-2-carbonsäurederivate 4a, 5 und 6, deren Darstellung beschrieben wird, liefern bei der Umsetzung nach einer Variante der Polonovski-Reaktion unterschiedliche Resultate. Aus 4a werden neben 9 der Ester 7 sowie 8 erhalten, w...

On the reaction of 2??chloroethylisothiocyanate with aromatic amines

: Outcalt, Russell J. Journal of Heterocyclic Chemistry, 1987 , vol. 24, p. 1425 - 1428

Abstract The reaction of aromatic amines with 2-chloroethylisothiocyanate 2 to give 2- arylaminothiazolines 1 was investigated. The course of this reaction was found to depend on the electronic nature of the amine and the reaction conditions. With arylamines ...

Aminopyrazoles. IV. Pyrazol??3??and 5??amines from 2, 3??dihaloalkanenitriles or 3??chloroacrylonitriles and hydrazines

: Ege, Guenter; Franz, Hermann Journal of Heterocyclic Chemistry, 1982 , vol. 19, p. 1267 - 1273

Nov-Dec 1982 Aminopyrazoles. IV. 1269 Table Preparation of Pyrazol-3-amines 4 and (or) -5-amines 5 4 Í3-NH, 64 65.5 (130/0.6) 211 (a) 11.5 88-89 160 (a) 84 65.5-68 (98/3) 4,5 R' R4 R5 in 4 or Method Yield Mp (°С) 'H NMR (deuteriochloroform) Kef R3 in 5 % (Ьр/...