常用名 | ADAMTS-5 inhibitor 8 | CAS号 | 1394122-20-3 |
---|---|---|---|
价格 | ¥需询单/100mg ¥需询单/250mg ¥需询单/1g | 纯度 | 98.0% |
备货期 | 10天 | 库存 | 现货 |
产品详情(用途,包装等)
用途: ADAMTS-5 inhibitor 8 is a highly potent and selective inhibitor of metalloprotease ADAMTS-5 with IC50 of 30 nM, >50-fold selectivity against ADAMTS-4 and >1000-fold selectivity against ADAMTS-1/13, MMP-13 and TACE; inhibits aggrecanase-mediated (374)ARGS neoepitope release from aggrecan and glycosaminoglycan in response to IL-1β/OSM stimulation. 物理化学性质: CAS号:1394122-20-3 常用中文名:ADAMTS-5 inhibitor 8 常用英文名:ADAMTS-5 inhibitor 8 分子式:C29H36N8O2S3 分子量:624.844 密度:1.3±0.1 g/cm3 沸点:821.9±75.0 °C at 760 mmHg 熔点:N/A 闪点:450.8±37.1 °C |