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Rv1625c agonist V-59

更新时间:2024-07-17 16:20:32 采购访问:14次

常用名 Rv1625c agonist V-59 CAS号 958588-17-5
价格 ¥需询单/100mg ¥需询单/250mg ¥需询单/1g 纯度 98.0%
备货期 10天 库存 现货
 产品详情(用途,包装等)
用途:
Rv1625c agonist V-59 (V-59) is a specific small molecule agonist of the Mtb adenylyl cyclase Rv1625c, inhibits Mtb growth in macrophages (EC50=0.3 uM) in an Rv1625c-dependent mechanism.V-59 inhibits Mtb growth in cholesterol media (EC50 0.70 uM), but not in media containing the two-carbon fatty acid acetate, or in standard rich growth media.V-59 stimulates Rv1625c to produce cAMP, which is necessary for V-59 to inhibit Mtb growth.Chemically activating Rv1625c via V-59 preferentially inhibits cholesterol utilization in WT Mtb, rather than equally inhibiting all lipid utilization by the bacterium.
物理化学性质:
CAS号:958588-17-5
常用中文名:Rv1625c agonist V-59
常用英文名:Rv1625c agonist V-59
分子式:C17H18FN7O2
分子量:371.376
密度:N/A
沸点:N/A
熔点:N/A
闪点:N/A

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