| 常用名 | PKI-179 hydrochloride | CAS号 | 1463510-35-1 |
|---|---|---|---|
| 价格 | 纯度 | 98.0% | |
| 备货期 | 10天 | 库存 | 现货 |
| 产品详情(用途,包装等)
用途: PKI-179 hydrochloride is a potent and orally active dual PI3K/mTOR inhibitor, with IC50s of 8 nM, 24 nM, 74 nM, 77 nM, and 0.42 nM for PI3K-α, PI3K-β, PI3K-γ, PI3K-δ and mTOR, respectively. PKI-179 hydrochloride also exhibits activity over E545K and H1047R, with IC50s of 14 nM and 11 nM, respectively. PKI-179 hydrochloride shows anti-tumor activity in vivo[1][2]. 物理化学性质: CAS号:1463510-35-1 常用中文名:PKI-179 hydrochloride 常用英文名:PKI-179 hydrochloride 分子式:C25H29ClN8O3 分子量:525.00 密度:N/A 沸点:N/A 熔点:N/A 闪点:N/A |