| 常用名 | PF-06679142 | CAS号 | 1467059-66-0 |
|---|---|---|---|
| 价格 | ¥需询单/1mg | 纯度 | 98.0% |
| 备货期 | 1天 | 库存 | 询单 |
| 产品详情(用途,包装等)
用途: PF-06679142 is a novel potent, orally active, α1β1γ1/α2β1γ1-isoform selective AMPK activator with Kd of 14 nM, EC50 of 22 nM for α1β1γ1-AMPK, shows minimal activity at the β2-containing isoforms (α1β2γ1, α2β2γ1, α2β2γ3); demonstrates in vivo target engagement experiment in ZSF-1 rats, an obese/diabetic rodent model of diabetic nephropathy. 物理化学性质: CAS号:1467059-66-0 常用中文名:PF-06679142 常用英文名:PF-06679142 分子式:C20H17F2NO3 分子量:357.357 密度:N/A 沸点:N/A 熔点:N/A 闪点:N/A |