常用名 | Cl-amidine TFA | CAS号 | 1043444-18-3 |
---|---|---|---|
价格 | ¥需询单/1g ¥需询单/1mg | 纯度 | 98.0% |
备货期 | 需询单 | 库存 | 询单 |
产品详情(用途,包装等)
用途: Cl-amidine TFA is an orally active peptidylarginine deminase (PAD) inhibitor, with IC50 values of 0.8 μM, 6.2 μM and 5.9 μM for PAD1, PAD3, and PAD4, respectively. Cl-amidine TFA induces apoptosis in cancer cells. Cl-amidine TFA induces microRNA (miR)-16 expression and causes cell cycle arrest. Cl-Amidine TFA prevents histone 3 citrullination and neutrophil extracellular trap formation, and improves survival in a murine sepsis model[1][2][3][4][5]. 物理化学性质: CAS号:1043444-18-3 常用中文名:Cl-amidine TFA 常用英文名:Cl-amidine TFA 分子式:C16H20ClF3N4O4 分子量:424.803 密度:N/A 沸点:N/A 熔点:N/A 闪点:N/A 储存条件:-20℃ |