| 常用名 | CA-4948 | CAS号 | 1801343-74-7 |
|---|---|---|---|
| 价格 | ¥1000.0/1g | 纯度 | 98.0% |
| 备货期 | 3天 | 库存 | 现货 |
| 产品详情(用途,包装等)
Product Name:CA-4948 CAS:1801343-74-7 MF:C21H19N7O3 Package:1g/bottle 一种可逆性激酶抑制剂,在TLR和IL-1R信号级联反应中,调节IRAK4的功能。在体内外实验中,具有良好的药代动力学特征和抗肿瘤活性。CA-4948isapotent,andorallyactiveinterleukin-1receptor-associatedkinase4(IRAK4)inhibitor.CA-4948exhibitedthegreatestefficacyinfourofthefiveABC-DLBChemicalbookCLPDXmodelstestedascomparedtoGBC-DLBCLandABC/GCBDLBCLPDXmodels.Furthermore,CA-4948wasefficaciousinABC-DLBCLPDXtumorscontainingactivatingmutationsinbothTLR/IL-1RandBCRsignalingpathways(MYD88andCD79Bdoublemutants). |