| 常用名 | GPR183 antagonist SAE-14 | CAS号 | 1241280-25-0 |
|---|---|---|---|
| 价格 | ¥1000.0/10mg | 纯度 | 98.6% |
| 备货期 | 需询单 | 库存 | 询单 |
| 产品详情(用途,包装等)
用途: GPR183 antagonist SAE-14 is a potent, selective GPR183 antagonist with IC50 of 28.5 nM, inhibits GPR183-dependent 7α,25-dihydroxycholesterol-induced calcium signaling in HL-60 cells.GPR183 antagonist SAE-14 inhibits calcium mobilization induced by 7α,25-OHC (EC80 209 nM).GPR183 antagonist SAE-14 reversed CCI-induced mechanical allodynia in a time-dependent manner when administered in vivo to mice.7α,25-dihydroxycholesterol induced allodynia in mice, SAE-14 blocked the effects of 7α,25-OHC in a dose-dependent manner. 物理化学性质: CAS号:1241280-25-0 常用中文名:GPR183 antagonist SAE-14 常用英文名:GPR183 antagonist SAE-14 分子式:C19H19F3N2O2 分子量:364.368 密度:N/A 沸点:N/A 熔点:N/A 闪点:N/A |