常用名 | Samuraciclib | CAS号 | 1805833-75-3 |
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价格 | ¥950.0/100mg ¥1700.0/250mg ¥3600.0/1g | 纯度 | 98.0% |
备货期 | 1天 | 库存 | 3 |
产品网页 | https://www.dcchemicals.com/product_show-samuraciclib.html |
产品详情(用途,包装等)
Samuraciclib (CT7001) is a potent, selective, ATP-competitive and orally active CDK7 inhibitor, with an IC50 of 41 nM. Samuraciclib displays 45-, 15-, 230- and 30-fold selectivity over CDK1, CDK2 (IC50 of 578 nM), CDK5 and CDK9, respectively. Samuraciclib inhibits the growth of breast cancer cell lines with GI50 values between 0.2-0.3 µM. Samuraciclib has anti-tumor effects. |