常用名 | LY2795050 | CAS号 | 1346133-08-1 |
---|---|---|---|
价格 | $需询单/100g $需询单/1kg $需询单/100kg $需询单/1000kg | 纯度 | 98.0% |
备货期 | 需询单 | 库存 | 询单 |
产品详情(用途,包装等)
用途: LY2795050 is a novel selective κ-opioid Receptor (KOR) antagonist (IC50=0.72 nM) and has the potential as a PET tracer to image KOR in vivo.IC50 Value: 0.72 nM (κ-opioid Receptor); 25.8 nM (κ-opioid) [1]Target: κ-opioid Receptorin vitro: LY2795050 displays full antagonist activity and high binding affinity and selectivity for KOR with a ki value of 0.72 nM [1].in vivo: In the brain, (11)C-LY2795050 displayed fast uptake kinetics (regional activity peak times of 物理化学性质: CAS号:1346133-08-1 常用中文名:LY2795050 常用英文名:LY2795050 分子式:C23H22ClN3O2 分子量:407.89300 密度:N/A 沸点:N/A 熔点:N/A 闪点:N/A 储存条件:2-8℃ |