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ELACRIDAR HYDROCHLORIDE

更新时间:2021-07-26 18:31:54 采购访问:53次

常用名 依克立达盐酸盐 CAS号 143851-98-3
价格 $需询单/100g $需询单/1kg $需询单/100kg $需询单/1000kg 纯度 98.0%
备货期 需询单 库存 询单
 产品详情(用途,包装等)
用途:
Elacridar Hcl (GF120918; GW0918) is a P-glycoprotein inhibitor, and has been used both in vitro and in vivo as a tool inhibitor of P-glycoprotein (Pgp) to investigate the role of transporters in the disposition of various test molecules.IC50 value:Target: P-glycoprotein In vitro, GF120918A demonstrated high plasma protein binding across species, although a definitive protein binding evaluation was precluded by poor recovery, particularly in buffer and in mouse, rat, and dog plasma. GF120918A did not demonstrate potent inhibition of several human cytochrome P450 enzymes evaluated in vitro, with IC(50) values well above concentrations anticipated to be achieved in vivo. Together, these data confirm the utility of GF120918A as a tool P-glycoprotein inhibitor in preclinical species and offer additional guidance on preclinical dose regimens likely to produce P-glycoprotein-mediated effects.
物理化学性质:
CAS号:143851-98-3
常用中文名:依克立达盐酸盐
常用英文名:Elacridar hydrochloride
分子式:C34H34ClN3O5
分子量:600.10400
密度:N/A
沸点:701.6ºC at 760 mmHg
熔点:N/A
闪点:378.1ºC
储存条件:2-8℃

供应商信息

达阳化工(杭州)有限公司 认证供应商

认证状态:已认证供应商
商品数:50181件
电话:+86571-88938639
地址:浙江省杭州市西湖区文三路259号2栋9楼
地区: 浙江省 杭州市 西湖区
联系人:王小姐
联系人电话:+86-571-8893-8639
邮件:enquiry@dycnchem.com
网址:http://www.dycnchem.com
主要市场:Mainly in Southeast Asia and European and American markets
年贸易额:10 to 20 million USD
外贸占销售比例:90%
主要合作伙伴:
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参考价格:$91/10mg
其他供应商价格:
2022-11-29 Elacridar hydrochloride
价格:¥需询单
2022-02-19 Elacridar hydrochloride
价格:¥476.9
2018-10-30 依克立达盐酸盐
价格:¥需询单
2021-02-06 Elacridar hydrochloride
价格:¥1707.0
2021-05-10 依克立达盐酸盐
价格:¥需询单
2022-05-12 Elacridar HCl
价格:$需询单

查看所有价格,请点击依克立达盐酸盐价格