| 常用名 | 5-[4-氟-1-[(6-甲基-2-吡啶基)乙酰基]-2,3-二氢-1H-吲哚-5-基]-7-甲基-7H-吡咯并[2,3-d]嘧啶-4-胺 | CAS号 | 1337532-29-2 |
|---|---|---|---|
| 价格 | $450.0/100mg $900.0/250mg $1900.0/1g $150.0/10ml | 纯度 | 98.0% |
| 备货期 | 3天 | 库存 | 3 |
| 产品网页 | https://www.dcchemicals.com/product_show-GSK2656157.html | ||
| 产品详情(用途,包装等)
GSK2656157 is an ATP-competitive inhibitor of PERK enzyme activity with an IC50 of 0.9 nM. It is highly selective for PERK with IC50 values >100 nM against a panel of 300 kinases. |