常用名 | 盐酸氯米帕明 | CAS号 | 17321-77-6 |
---|---|---|---|
价格 | ¥需询单/1kg | 纯度 | 98.0% |
备货期 | 需询单 | 库存 | 现货 |
产品详情(用途,包装等)
用途: Clomipramine HCl is a serotonin transporter (SERT), norepinephrine transporter (NET) dopamine transporter (DAT) blocker with Ki of 0.14, 54 and 3 nM, respectively. Target: 5-HT ReceptorClomipramine hydrochloride (Anafranil) is a hydrochloride salt of clomipramine which is a serotonin transporter (SERT), norepinephrine transporter (NET) dopamine transporter (DAT) blocker with Ki of 0.14, 54 and 3 nM, respectively. Clomipramine hydrochloride (Anafranil) is a tricyclic antidepressant. Clomipramine hydrochloride (Anafranil) is a norepinephrine-reuptake inhibitor and is an antiobsessional drug. Clomipramine hydrochloride (Anafranil) is an antagonist/inverse agonist at the following receptors: D2 receptor (Ki = 162 nM), D3 receptor (Ki = 30 nM), α1-adrenergic receptor (Ki = 3.2 nM), α2-adrenergic receptor (Ki = 525 nM), H1 receptor (Ki = 31 nM), mACh receptors (Ki = 37 nM), 5-HT2A receptor (Ki = 36 nM), 5-HT2C receptor (Ki = 65 nM), 5-HT3 receptor (Ki = 85 nM), 5-HT6 receptor (Ki = 54 nM), 5-HT7 receptor (Ki = 127 nM), D1 receptor (Ki = 219 nM) [1-3]. 物理化学性质: CAS号:17321-77-6 常用中文名:盐酸氯米帕明 常用英文名:Clomipramine HCl 分子式:C19H24Cl2N2 分子量:351.313 密度:N/A 沸点:434.2ºC at 760 mmHg 熔点:189-190°C 闪点:216.4ºC 储存条件:库房低温通风干燥,与食品原料分开存放 |