常用名 | 甲磺酸卡莫司他 | CAS号 | 59721-29-8 |
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价格 | ¥需询单/10g | 纯度 | 95.0% |
备货期 | 14天 | 库存 | 咨询 |
产品详情(用途,包装等)
用途: Camostat Mesylate(FOY305; FOY-S980) is a trypsin-like protease inhibitorTarget: Trypsin-like proteaseCamostat mesilate (500 mM) inhibits generation of TGF-beta by suppressing plasmin activity and reduces the activity of TGF-beta, which blocks in vitro activation of HSCs [1]. Camostat mesilate (20 mM) combined with insulin results a significant hypoglycemic effect following large intestinal administration. Camostat mesilate (20 mM) is effective in reducing insulin degradation in both small and large intestinal homogenates of rats [2]. Camostat mesilate (2 mM) inhibits MCP-1 and TNF- production in activated rat monocytes. Camostat mesilate (2 mM) inhibits proliferation and MCP-1 production of cultured rat PSCs. Camostat mesilate (1 mg/g) prevents pancreatic atrophy and improves pancreatic exocrine function of rat chronic pancreatitis induced by DBTC. Camostat mesilate (1 mg/g) inhibits chronic inflammation and pancreatic fibrosis induced by DBTC. Camostat mesilate (1 mg/g) inhibits the development of pancreatic fibrosis and PSCs activation in the pancreas induced by DBTC. Camostat mesilate (1 mg/g) suppresses monocytes infiltration and inhibits MCP-1 expression both in serum and in pancreatic tissue [3]. 物理化学性质: CAS号:59721-29-8 常用中文名:甲磺酸卡莫司他 常用英文名:Camostat Mesylate 分子式:C21H26N4O8S 分子量:494.518 密度:N/A 沸点:634.6ºC at 760 mmHg 熔点:150-1550C 闪点:N/A 储存条件:Desiccate at RT |