Affinity labels for. beta.-adrenoceptors: preparation and properties of alkylating. beta.-blockers derived from indole

…, W Buchowiecki, J Milecki, JW Kusiak

文献索引：Pitha, Josef; Buchowiecki, Wieslaw; Milecki, Jan; Kusiak, John W. Journal of Medicinal Chemistry, 1987 , vol. 30, # 4 p. 612 - 615

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被引用次数: 21

摘要

Results Chemistry. Reaction of (2)-1, 8-diamino-p-menthane (1) with epoxides 2 or 3 yielded mixtures from which the desired monosubstituted products were isolated; these obviously were mixtures of isomers (pair 4 and 5 and pair 6 and 7), but no suitable separation system could be found