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Discovery of 1, 5-benzodiazepines with peripheral cholecystokinin (CCK-A) receptor agonist activity (II): Optimization of the C3 amino substituent

GC Hirst, C Aquino, L Birkemo, DK Croom…

文献索引:Journal of Medicinal Chemistry, , vol. 39, # 26 p. 5236 - 5245

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被引用次数: 39

摘要

... Journal of Medicinal Chemistry. ... Departments of Medicinal Chemistry, Cellular Biochemistry, and Pharmacology, Glaxo Wellcome Research and Development, 5 Moore Drive, Research Triangle Park, North Carolina 27709. J. Med. Chem. ... Chemistry. ...