Receptor activity and conformational analysis of 5′-halogenated resiniferatoxin analogs as TRPV1 ligands

KS Lim, DW Kang, YS Kim, MS Kim, SG Park…

文献索引：Bioorganic and Medicinal Chemistry Letters, , vol. 21, # 1 p. 299 - 302

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被引用次数: 5

摘要

... Bioorganic & Medicinal Chemistry Letters. ... In this Letter, we have investigated the effect of halogenation in the A-region of RTX and of the isosteric 4-amino surrogate in a systematic manner and we describe the synthesis and receptor activity, as well as conformational analysis ...