Intramolecular inverse-electron-demand Diels-Alder reactions of imidazoles with 1, 2, 4-triazines: a new route to 1, 2, 3, 4-tetrahydro-1, 5-naphthyridines and related …

BR Lahue, SM Lo, ZK Wan, GHC Woo…

文献索引：Barlin, Gordon B.; Ireland, Stephen J.; Nguyen, Trang M. T.; Kotecka, Barbara; Rieckmann, Karl H. Australian Journal of Chemistry, 1994 , vol. 47, # 6 p. 1143 - 1154

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被引用次数: 53

摘要

... J. Org. ... cycloadditions employing a tetramethylene tether also proceeded to give 2,3,4,5-tetrahydro- 1H-pyrido[3,2-b]azepines in ... discovery as potential antimalarial candidates, 6b,12 ultimately evolving into large antimalarial programs as exemplified by the work of Barlin and co ...