Tetrahedron

The synthesis of N-arylcyclopropylamines via palladium-catalyzed C–N bond formation

W Cui, RN Loeppky

文献索引：Cui, Wenge; Loeppky, Richard N Tetrahedron, 2001 , vol. 57, # 15 p. 2953 - 2956

全文：HTML全文

被引用次数: 26

摘要

A variety of N-arylcyclopropylamines has been prepared in one step, by the Pd2 (dba) 3/BINAP/NaOtBu-catalyzed amination of an aryl bromide with cyclopropylamine. Compounds bearing the N-aryl substitutent (phenyl, 4-methylphenyl, 2-methoxyphenyl, 3-