Phosphonyltriethylammonium salts: novel reactive species for the synthesis of phosphonate esters and phosphonamides

…, W Moore, PA Sprengeler, J Witherington…

文献索引：Hirschmann, Ralph; Yager, Kraig M.; Taylor, Carol M.; Moore, William; Sprengeler, Paul A.; Witherington, Jason; Phillips, Barton W.; Smith III, Amos B. Journal of the American Chemical Society, 1995 , vol. 117, # 23 p. 6370 - 6371

全文：HTML全文

被引用次数: 28

摘要

Phosphonate esters and amides find great utility as stable mimetics of tetrahedral transition states. Transition state analogs incorporating these functionalities have been exploited inter alia as enzyme inhibitors' and as haptens for catalytic antibody research,* including the recently reported formation of dipeptide~.~ Phosphonate esters and phosphonamides are generally prepared by the reaction of phosphonochloridates or phosphonodi~ hloridates~ ...