Synthesis and Biological Evaluation of Dihydroisoquinoline-2 (1H)-Carbothioamide Derivatives as TRPV1 Antagonists

H Qian, W Chen, X Zhang, H Zhang…

文献索引：Letters in Drug Design and Discovery, , vol. 7, # 4 p. 235 - 237

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摘要

... Its antagonists are expected to prevent pain perception by blocking the receptor directly. In this letter, eight dihydroisoquinoline-2(1H)-carbothioamide derivatives were designed and synthesized as TRPV1 antagonists. ... 236 Letters in Drug Design & Discovery, 2010, Vol. ...