Palladium??Catalyzed Direct and Site??Selective Desulfitative Arylation of Indoles with Sodium Sulfinates

…, J Luo, F Xiao, S Zhang, GJ Deng…

文献索引：Wu, Mingyue; Luo, Jiaying; Xiao, Fuhong; Zhang, Shufeng; Deng, Guo-Jun; Luo, He-An Advanced Synthesis and Catalysis, 2012 , vol. 354, # 2-3 p. 335 - 340

全文：HTML全文

被引用次数: 77

摘要

Abstract An efficient method was developed for the desulfitative arylation of indoles with sodium sulfinates using palladium as catalyst and copper chloride dihydrate as oxidant. The direct arylation occurred exclusively in the C-2 position of indoles and proceeded well for a range of different substrates.