Application of Sharpless asymmetric dihydroxylation to thienyl-and benzothienyl acrylates and crotonates

…, M De Bonis, M Funicello, P Lupattelli, R Pandolfo

文献索引：Bonini, Carlo; Chiummiento, Lucia; De Bonis, Margherita; Funicello, Maria; Lupattelli, Paolo; Pandolfo, Rocco Tetrahedron Asymmetry, 2006 , vol. 17, # 20 p. 2919 - 2924

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被引用次数: 14

摘要

Optimized conditions for the catalytic asymmetric dihydroxylation have been applied to thiophene and benzothiophene containing acrylates and crotonates to afford the corresponding diols in good overall yields and good to excellent enantiomeric excess. The products obtained were revealed to be useful intermediates in peptidomimetic synthesis.