N′-3-(Trifluoromethyl) phenyl Derivatives of N-Aryl-N′-methylguanidines as Prospective PET Radioligands for the Open Channel of the N-Methyl-d-aspartate ( …
... Volume: Page: ... For example, 7 was obtained by treating 1-naphthylamine hydrochloride with N-methyl-N-(3-(trifluoromethyl)phenyl)cyanamide at 130 °C in ... Usually, if the inhibition exceeded ∼89%, a K i value was determined, also with [ 3 H]TCP as radioligand ...