Access to 3??Arylindoles through a Tandem One??Pot Protocol Involving Dearomatization, a Regioselective Michael Addition Reaction, and Rearomatization

…, S Putturu, R Kuppusamy, KC Boellaard…

文献索引：Chittimalla, Santhosh Kumar; Bandi, Chennakesavulu; Putturu, Sireesha; Kuppusamy, Rajesh; Boellaard, Kevin Christopher; Tan, David Chu Aan; Lum, Demi Ming Jie European Journal of Organic Chemistry, 2014 , vol. 2014, # 12 p. 2565 - 2575

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被引用次数: 6

摘要

Abstract A facile, general and rapid protocol for the introduction of oxygenated aryls at the 3- position of indoles is described. This approach consists of a tandem dearomatization, a regioselective Michael addition reaction, and rearomatization in a one-pot three-step sequence to obtain 3-arylindoles in good yields.