Acetamide Scanning around Bicyclic Thiazoles: SAR at the H3 Receptor

F Denonne, S Célanire, B Christophe…

文献索引：ChemMedChem, , vol. 6, # 9 p. 1559 - 1565

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被引用次数: 2

摘要

... ChemMedChem, 6: 1559–1565. ... Volume: Issue: Page ... c) 3, DMF, 60 °C, 2 h (83 %); d) MsCl, Et 3 N, CH 2 Cl 2 , 20 °C, 12 h, (92 %); e) p-HOPhCO 2 H, HBr/AcOH, 20 °C, 5 days (9 %); f) AcCl, Et 3 N, CH 2 Cl 2 , 20 °C, 2 h, (55 %); g) 2-methylpyrrolidine, CH 3 CN, 100 °C, 6 h, (33 ...