Synthesis of Linear Aza and Thio Analogues of Acetogenins and Evaluation of Their Cytotoxicity

P Villo, L Toom, E Eriste, L Vares

文献索引：Villo, Piret; Toom, Lauri; Eriste, Elo; Vares, Lauri European Journal of Organic Chemistry, 2013 , # 30 p. 6886 - 6899

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被引用次数: 1

摘要

Abstract We report the stereoselective synthesis of thio and aza analogues of Annonaceous acetogenins. The synthetic route allows easy variation of the stereochemistry and of the thio- and aza-fragments. Kinetic resolution of terminal bis-epoxides was used to set two remote ...