The synthesis of novel GABA uptake inhibitors. 1. Elucidation of the structure-activity studies leading to the choice of (R)-1-[4, 4-bis (3-methyl-2-thienyl)-3-butenyl]-3- …

KE Andersen, C Braestrup, FC Groenwald…

文献索引：Journal of Medicinal Chemistry, , vol. 36, # 12 p. 1716 - 1725

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被引用次数: 121

摘要

... CI-966 has been in- vestigated in a phase I clinical trial.w We wish to report the synthesis" and biological activity of a series of novel and selective GABA uptake inhibitors 0 1993 American Chemical Society ... Page 3. 1718 Journal of Medicinal Chemistry, 1993, Vol. ...