文献索引：Hagedorn, Alfred A.; Erhardt, Paul W.; Lumma, William C.; Wohl, Ronald, A.; Cantor, Elinor; et al. Journal of Medicinal Chemistry, 1987 , vol. 30, # 8 p. 1342 - 1347
As shown in Scheme 11, an alternative synthesis was employed for the imidazol-2-yl compounds 9r and 98, the meta-substituted example 9t, and the imidazolylmethyl compound 9v. These were prepared by acylation of 10 with the imidazolylbenzoic acids 12, again in PPA or, preferably, Eaton's acid. This procedure is also applicable to the preparation of the p- imidazol-1-yl compounds and, when optimized, is well suited for large-scale preparations. ...
