Tetrahedron

One-pot aromatic amination based on carbon–nitrogen coupling reaction between aryl halides and azido compounds

…, Y Shimoda, K Nozaki, S Mori, Y Sawama, Y Monguchi…

文献索引：Maejima, Toshihide; Shimoda, Yutaka; Nozaki, Kei; Mori, Shigeki; Sawama, Yoshinari; Monguchi, Yasunari; Sajiki, Hironao Tetrahedron, 2012 , vol. 68, # 6 p. 1712 - 1722

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被引用次数: 28

摘要

An efficient copper-mediated C–N coupling reaction between various aryl halides and azido compounds to produce the corresponding aromatic primary amines was established. The present amination is apparently involved in both the reduction of an azido functionality to the corresponding primary amino group and its cross-coupling reaction with aryl halides in a one-pot manner. The present amination could be applied to the synthesis of procaine, a ...