Process Development of a Novel Azetidinyl Ketolide Antibiotic

B Li, TV Magee, RA Buzon, DW Widlicka…

文献索引：Organic Process Research and Development, , vol. 16, # 5 p. 788 - 797

被引用次数: 3

摘要

... bacterial pneumonia (CABP) and biodefense pathogens.(5) Efforts in our antibacterial research program led to ... The process efficiency could be greatly improved by telescoping the steps. ... an aqueous workup for the acetylation step was still needed, the organic phase could be ...

50720-12-2

3-溴-5-甲氧基吡啶

342603-10-5

3-BOC-氨基-5-甲氧基吡啶

Synthesis of a 5-alkoxypyrido [3, 4-d] pyrimidin-4 (3H)-one ...

[Dishington, Allan P.; Johnson, Paul D.; Kettle, Jason G. Tetrahedron Letters, 2004 , vol. 45, # 19 p. 3733 - 3735]

Synthesis of a 5-alkoxypyrido [3, 4-d] pyrimidin-4 (3H)-one ...

[Tetrahedron Letters, , vol. 45, # 19 p. 3733 - 3735]

Process Development of a Novel Azetidinyl Ketolide Antibioti...

[Li, Bryan; Magee, Thomas V.; Buzon, Richard A.; Widlicka, Daniel W.; Bill, Dave R.; Brandt, Thomas; Cao, Xiaoping; Coutant, Michael; Dou, Haijian; Granskog, Karl; Flanagan, Mark E.; Hayward, Cheryl M.; Li, Bin; Liu, Fengwei; Liu, Wei; Nguyen, Thuy-Trinh; Raggon, Jeffrey W.; Rose, Peter; Rainville, Joseph; Reilly, Usa Datta; Shen, Yue; Sun, Jianmin; Wilcox, Glenn E. Organic Process Research and Development, 2012 , vol. 16, # 5 p. 788 - 797]