Guanidinum Chloride as Dehydrocyclization Agent in the Synthesis of 2??Fuctionalized (4H)??3, 1??Benzoxazine??4??ones

…, F Havasi, M Sharafi??Kolkeshvandi

文献索引：Nikpour, Farzad; Bahmani, Asrin; Havasi, Forugh; Sharafi-Kolkeshvandi, Mahnaz Journal of Heterocyclic Chemistry, 2014 , vol. 51, # 1 p. 34 - 37

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摘要

Abstract A facile and expedient route for the synthesis of 2-ethoxy-and 2-(ethylcarboxylate)- (4H)-3, 1-benzoxazine-4-ones is described using guanidinium chloride as a safe and convenient dehydrocyclization agent. High yields of the products obtain under mild reaction conditions without need to use of any catalyst and with easy work-up of the reaction mixture.